Per Artursson
Active 1984–2024
- 147
- Papers
- 28,836
- Citations
- 96
- h-index
- 142
- i10-index
Citations
Citation sources
Countries
Institutions
Fields
- Medicine28.3%
- Biochemistry, Genetics and Molecular Biology21%
- Pharmacology, Toxicology and Pharmaceutics19.9%
- Computer Science8.8%
- Materials Science4.6%
- Chemistry3.5%
- Other13.9%
Topics
- Drug Transport and Resistance Mechanisms6.9%
- Advanced Drug Delivery Systems6.6%
- Computational Drug Discovery Methods4.8%
- Drug Solubulity and Delivery Systems4.4%
- RNA Interference and Gene Delivery3.1%
- Pharmacogenetics and Drug Metabolism2.5%
- Other71.7%
Coauthors
- Christel A. S. Bergström15
- Kristina Luthman15
- Pär Matsson15
- Christine Wegler13
- Ulf Norinder13
- Jacek R. Wiśniewski11
- Johan Karlsson10
- Tommy B. Andersson9
- Anders Åsberg8
- Anna‐Lena Ungell8
- Jøran Hjelmesæth8
- Niklas Handin8
- Patric Stenberg8
- André Mateus7
- Hege Christensen7
- Ida Robertsen7
- Katrin Palm7
- Kjell M. Vårum7
- Lucia Lazorova7
- Maria Karlgren7
- Alex Avdeef6
- Gustav Ahlin6
- Hans Lennernäs6
- Johan Gråsjö6
All papers
- Determination of drug permeability and prediction of drug absorption in Caco-2 monolayers
Authors: Ina Hubatsch, Eva Ragnarsson, Per Artursson - Nature Protocols 2007 cited by 1,458
- Oral absorption of peptides and nanoparticles across the human intestine: Opportunities, limitations and studies in human tissues
Authors: Patrik Lundquist, Per Artursson - Advanced Drug Delivery Reviews 2016 cited by 476
- Caco-2 monolayers in experimental and theoretical predictions of drug transport1PII of original article: S0169-409X(96)00415-2. The article was originally published in Advanced Drug Delivery Reviews 22 (1996) 67–84.1
Authors: Per Artursson, Katrin Palm, Kristina Luthman - Advanced Drug Delivery Reviews 2001 cited by 1,534
- Correlation between oral drug absorption in humans and apparent drug permeability coefficients in human intestinal epithelial (Caco-2) cells
Authors: Per Artursson, Johan Karlsson - Biochemical and Biophysical Research Communications 1991 cited by 1,868
- MTH1 inhibition eradicates cancer by preventing sanitation of the dNTP pool
Authors: Helge Gad, Tobias Koolmeister, Ann‐Sofie Jemth, Saeed Eshtad, Sylvain A. Jacques, Cecilia Ström, L. Svensson, Niklas Schultz, Thomas Lundbäck, Berglind O. Einarsdottir, Aljona Saleh, Camilla Göktürk, Paweł Baranczewski, Richard Svensson, Ronnie P.‐A. Berntsson, Robert Gustafsson, Kia Strömberg, Kumar Sanjiv, Marie‐Caroline Jacques‐Cordonnier, Matthieu Desroses, Anna‐Lena Gustavsson, Roger Olofsson Bagge, Fredrik Johansson, Evert Homan, Olga Loseva, Lars Bräutigam, L. E. B. Johansson, Andreas Höglund, Anna Hagenkort, Therese Pham, Mikael Altun, Fabienne Z. Gaugaz, Svante Vikingsson, Bastiaan Evers, Martin Henriksson, Karl S. A. Vallin, Olov Wallner, Lars G.J. Hammarström, Elisée Wiita, Ingrid Almlöf, Christina Kalderén, Hanna Axelsson, Tatjana Djureinovic, Jordi Carreras‐Puigvert, Maria Häggblad, Fredrik Jeppsson, Ulf Märtens, Cecilia Lundin, Bo Lundgren, Ingrid Granelli, Annika Jenmalm Jensen, Per Artursson, Jonas A. Nilsson, Pål Stenmark, Martin Scobie, Ulrika Warpman Berglund, Thomas Helleday - Nature 2014 cited by 529
- Small-molecule inhibitor of OGG1 suppresses proinflammatory gene expression and inflammation
Authors: Torkild Visnes, Armando Cázares‐Körner, Wenjing Hao, Olov Wallner, Geoffrey Masuyer, Olga Loseva, Oliver Mortusewicz, Elisée Wiita, Antonio Sarno, Aleksandr Manoilov, Juan Astorga‐Wells, Ann‐Sofie Jemth, Lang Pan, Kumar Sanjiv, Stella Karsten, Camilla Göktürk, Maurice Grube, Evert Homan, Bishoy Hanna, Cynthia B. J. Paulin, Therese Pham, Azita Rasti, Ulrika Warpman Berglund, Catharina Von Nicolai, Carlos Benitéz‐Buelga, Tobias Koolmeister, Dag Ivanic, Petar Iliev, Martin Scobie, Hans E. Krokan, Paweł Baranczewski, Per Artursson, Mikael Altun, Annika Jenmalm Jensen, Christina Kalderén, Xueqing Ba, Roman A. Zubarev, Pål Stenmark, István Boldogh, Thomas Helleday - Science 2018 cited by 233
- Coexistence of passive and carrier-mediated processes in drug transport
Authors: Kiyohiko Sugano, Manfred Kansy, Per Artursson, Alex Avdeef, Stefanie Bendels, Li Di, Gerhard F. Ecker, Bernard Faller, Holger Fischer, Grégori Gerebtzoff, Hans Lennernaes, Frank Senner - Nature Reviews Drug Discovery 2010 cited by 653
- Structural and conformational determinants of macrocycle cell permeability
Authors: Björn Over, Pär Matsson, Christian Tyrchan, Per Artursson, B.C. Doak, Michael A. Foley, Constanze Hilgendorf, Stephen Johnston, Maurice D. Lee, Richard J. Lewis, Patrick McCarren, Giovanni Muncipinto, Ulf Norinder, Matthew W. D. Perry, Jeremy R. Duvall, Jan Kihlberg - Nature Chemical Biology 2016 cited by 213
- Polar Molecular Surface Properties Predict the Intestinal Absorption of Drugs in Humans
Authors: Katrin Palm, Patric Stenberg, Kristina Luthman, Per Artursson - Pharmaceutical Research 1997 cited by 751
- The Critical Role of Passive Permeability in Designing Successful Drugs
Authors: Li Di, Per Artursson, Alex Avdeef, Leslie Z. Benet, J. Brian Houston, Manfred Kansy, Edward H. Kerns, Hans Lennernäs, Dennis A. Smith, Kiyohiko Sugano - ChemMedChem 2020 cited by 109
- In-depth quantitative analysis and comparison of the human hepatocyte and hepatoma cell line HepG2 proteomes
Authors: Jacek R. Wiśniewski, Anna Vildhede, Agneta Norén, Per Artursson - Journal of Proteomics 2016 cited by 184
- Current challenges and future perspectives in oral absorption research: An opinion of the UNGAP network
Authors: Zahari Vinarov, Bertil Abrahamsson, Per Artursson, Hannah Batchelor, Philippe Berben, Andreas Bernkop‐Schnürch, James Butler, Jens Ceulemans, Nigel Davies, Didier Dupont, Gøril Eide Flaten, Nikoletta Fotaki, Brendan T. Griffin, Vincent Jannin, Janneke Keemink, Filippos Kesisoglou, Mirko Koziolek, Martin Kuentz, Alan R. Mackie, Antonio J. Meléndez‐Martínez, Mark McAllister, Anette Müllertz, Caitríona M. O’Driscoll, Neil Parrott, Jadwiga Paszkowska, Petr Pávek, Christopher J. H. Porter, Christos Reppas, Cordula Stillhart, Kiyohiko Sugano, Elena Toader, Kateřina Valentová, Maria Vertzoni, Saskia N. de Wildt, Clive Wilson, Patrick Augustijns - Advanced Drug Delivery Reviews 2021 cited by 145
- Expression of Thirty-six Drug Transporter Genes in Human Intestine, Liver, Kidney, and Organotypic Cell Lines
Authors: Constanze Hilgendorf, Gustav Ahlin, Annick Seithel, Per Artursson, Anna‐Lena Ungell, Johan Karlsson - Drug Metabolism and Disposition 2007 cited by 580
- Classification of Inhibitors of Hepatic Organic Anion Transporting Polypeptides (OATPs): Influence of Protein Expression on Drug–Drug Interactions
Authors: Maria Karlgren, Anna Vildhede, Ulf Norinder, Jacek R. Wiśniewski, Emi Kimoto, Yurong Lai, U Haglund, Per Artursson - Journal of Medicinal Chemistry 2012 cited by 365
- CETSA screening identifies known and novel thymidylate synthase inhibitors and slow intracellular activation of 5-fluorouracil
Authors: Helena Almqvist, Hanna Axelsson, Rozbeh Jafari, Dan Chen, André Mateus, Martin Haraldsson, Andreas Larsson, Daniel Martinez Molina, Per Artursson, Thomas Lundbäck, P. Nordlund - Nature Communications 2016 cited by 164
- Global variability analysis of mRNA and protein concentrations across and within human tissues
Authors: Christine Wegler, Magnus Ölander, Jacek R. Wiśniewski, Patrik Lundquist, Katharina Zettl, Anders Åsberg, Jøran Hjelmesæth, Tommy B. Andersson, Per Artursson - NAR Genomics and Bioinformatics 2019 cited by 103
- Hepatocyte size fractionation allows dissection of human liver zonation
Authors: Magnus Ölander, Christine Wegler, Inken Flörkemeier, Andrea Treyer, Niklas Handin, Jenny M. Pedersen, Anna Vildhede, André Mateus, Edward L. LeCluyse, Jozef Urdzik, Per Artursson - Journal of Cellular Physiology 2021 cited by 24
- Regional levels of drug transporters along the human intestinal tract: Co-expression of ABC and SLC transporters and comparison with Caco-2 cells
Authors: Gunilla Englund, Fredrik Rorsman, Anders Rönnblom, Urban Karlbom, Lucia Lazorova, Johan Gråsjö, Andreas Kindmark, Per Artursson - European Journal of Pharmaceutical Sciences 2006 cited by 368
- Absorption Enhancement through Intracellular Regulation of Tight Junction Permeability by Medium Chain Fatty Acids in Caco-2 Cells
Authors: Tuulikki Lindmark, Yukitaka Kimura, Per Artursson - Journal of Pharmacology and Experimental Therapeutics 1998 cited by 327
- Mechanisms of absorption enhancement by medium chain fatty acids in intestinal epithelial Caco-2 cell monolayers.
Authors: Tuulikki Lindmark, T Nikkilä, Per Artursson - Journal of Pharmacology and Experimental Therapeutics 1995 cited by 194
- Validation and development of MTH1 inhibitors for treatment of cancer
Authors: Ulrika Warpman Berglund, Kumar Sanjiv, Helge Gad, Christina Kalderén, Tobias Koolmeister, Therese Pham, Camilla Göktürk, Rozbeh Jafari, Gianluca Maddalo, Brinton Seashore‐Ludlow, Alexey Chernobrovkin, Aleksandr Manoilov, Ioannis S. Pateras, Azita Rasti, Ann‐Sofie Jemth, Ingrid Almlöf, Olga Loseva, Torkild Visnes, Berglind O. Einarsdottir, Fabienne Z. Gaugaz, Amyza Saleh, Björn Platzack, Olov Wallner, Karl S. A. Vallin, Martin Henriksson, Prasad B. Wakchaure, Sanjay R. Borhade, Patrick Herr, Yvonne Kallberg, Paweł Baranczewski, Evert Homan, Elisée Wiita, Varun Nagpal, Thomas Meijer, Nicolaas Schipper, Sean G. Rudd, Lars Bräutigam, Annika Lindqvist, Anne M. Filppula, Te‐Chang Lee, Per Artursson, Jonas A. Nilsson, Vassilis G. Gorgoulis, Janne Lehtiö, Roman A. Zubarev, Martin Scobie, Thomas Helleday - Annals of Oncology 2016 cited by 145
- Drug Disposition Protein Quantification in Matched Human Jejunum and Liver From Donors With Obesity
Authors: Christine Wegler, Jacek R. Wiśniewski, Ida Robertsen, Hege Christensen, Jens Kristoffer Hertel, Jøran Hjelmesæth, Rasmus Jansson‐Löfmark, Anders Åsberg, Tommy B. Andersson, Per Artursson - Clinical Pharmacology & Therapeutics 2022 cited by 41
- Effect of Chitosan on the Permeability of Monolayers of Intestinal Epithelial Cells (Caco-2)
Authors: Per Artursson, Tuulikki Lindmark, Stanley S. Davis, Lisbeth Illum - Pharmaceutical Research 1994 cited by 770
- Transport of Lipophilic Drug Molecules in a New Mucus-Secreting Cell Culture Model Based on HT29-MTX Cells
Authors: Isabel Behrens, Patric Stenberg, Per Artursson, Thomas Kissel - Pharmaceutical Research 2001 cited by 219
