Kenneth A. Jacobson
Active 1973–2025
- 304
- Papers
- 47,157
- Citations
- 114
- h-index
- 292
- i10-index
Citations
Citation sources
Countries
Institutions
Fields
- Biochemistry, Genetics and Molecular Biology58.2%
- Medicine20.3%
- Neuroscience8.2%
- Immunology and Microbiology3.1%
- Computer Science2.4%
- Chemistry1.8%
- Other6%
Topics
- Adenosine and Purinergic Signaling9.9%
- Receptor Mechanisms and Signaling5.3%
- Lipid Membrane Structure and Behavior4.2%
- Neuropeptides and Animal Physiology2.4%
- Neuroscience and Neuropharmacology Research2%
- Neuroinflammation and Neurodegeneration Mechanisms1.9%
- Other74.3%
Coauthors
- Zhan‐Guo Gao68
- Dilip K. Tosh28
- Daniela Salvemini23
- T. Kendall Harden21
- Christa E. Müller18
- Neli Melman17
- Xiao‐duo Ji17
- Gary L. Stiles15
- John W. Daly14
- José L. Boyer14
- Maria P. Abbracchio14
- Mark E. Olah13
- Veronica Salmaso13
- Zhoumou Chen13
- Stefano Moro12
- Yong‐Chul Kim12
- Bruce T. Liang11
- Kwan‐Young Jung11
- Geoffrey Burnstock10
- Raymond C. Stevens10
- Dag K.J.E. Von Lubitz9
- Shanu Jain9
- A. Michiel van Rhee8
- John A. Auchampach8
All papers
- Hematoxylin and Eosin Staining of Tissue and Cell Sections
Authors: Andrew H. Fischer, Kenneth A. Jacobson, Jack Rose, Rolf Zeller - Cold Spring Harbor Protocols 2008 cited by 2,113
- The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors
Authors: S P H Alexander, Arthur Christopoulos, Anthony P. Davenport, Eamonn Kelly, Alistair Mathie, John A. Peters, Emma L. Veale, Jane F Armstrong, Elena Faccenda, Simon D Harding, Jamie A. Davies, Maria P. Abbracchio, George Abraham, Alexander I. Agoulnik, Wayne Alexander, Khaled Alhosaini, Magnus Bäck, Jillian G. Baker, Nicholas M. Barnes, Ross A. D. Bathgate, Jean‐Martin Beaulieu, Annette G. Beck‐Sickinger, Maik Behrens, Kenneth E. Bernstein, Bernhard Bettler, N.J.M. Birdsall, Victoria A. Blaho, François Boulay, Corinne Bousquet, Hans Bräuner‐Osborne, Geoffrey Burnstock, Girolamo Calò, Justo P. Castaño, Kevin Catt, Stefania Ceruti, Paul L. Chazot, Nan Chiang, Bice Chini, Jerold Chun, Antonia Cianciulli, Olivier Civelli, Lucie H. Clapp, Réjean Couture, Helen M. Cox, Zsolt Csaba, Cláes Dahlgren, Gordon Dent, Steven D. Douglas, Pascal Dournaud, Satoru Eguchi, Emanuel Escher, Edward J. Filardo, Tung M. Fong, Marta Fumagalli, Raul R. Gainetdinov, Michael L. Garelja, Marc de Gasparo, Craig Gerard, Marvin C. Gershengorn, Fernand Gobeil, Theodore L. Goodfriend, Cyril Goudet, Lukas Grätz, Karen J. Gregory, Andrew L. Gundlach, Jörg Hamann, Julien Hanson, Richard L. Hauger, Debbie L. Hay, Ákos Heinemann, Deron R. Herr, Morley D. Hollenberg, Nicholas D. Holliday, Mastgugu Horiuchi, Daniël Hoyer, László Hunyady, Ahsan Husain, Adriaan P. IJzerman, Tadashi Inagami, Kenneth A. Jacobson, Robert T. Jensen, Ralf Jockers, Deepa Jonnalagadda, Sadashiva S. Karnik, Klemens Kaupmann, Jacqueline Kemp, Charles Kennedy, Yasuyuki Kihara, Takio Kitazawa, Paweł Kozielewicz, Hans‐Jürgen Kreienkamp, Jyrki P. Kukkonen, Tobias Langenhan, Dan Larhammar, Katie Leach, Davide Lecca, John D. Lee, Susan E. Leeman, Jérôme Leprince, Xaria X. Li and 66 more - British Journal of Pharmacology 2023 cited by 388
- UDP acting at P2Y6 receptors is a mediator of microglial phagocytosis
Authors: Schuichi Koizumi, Yukari Shigemoto‐Mogami, Kaoru Nasu‐Tada, Yoichi Shinozaki, Keiko Ohsawa, Makoto Tsuda, Bhalchandra V. Joshi, Kenneth A. Jacobson, Shinichi Kohsaka, Kazuhide Inoue - Nature 2007 cited by 815
- Update of P2X receptor properties and their pharmacology: IUPHAR Review 30
Authors: Péter Illés, Christa E. Müller, Kenneth A. Jacobson, Thomas Grütter, Annette Nicke, Samuel J. Fountain, Charles Kennedy, Günther Schmalzing, Michael F. Jarvis, Stanko S. Stojilković, Brian F. King, Francesco Di Virgilio - British Journal of Pharmacology 2020 cited by 310
- THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein‐coupled receptors
Authors: S P H Alexander, Arthur Christopoulos, Anthony P. Davenport, Eamonn Kelly, Alistair Mathie, John A. Peters, Emma L. Veale, Jane F Armstrong, Elena Faccenda, Simon D Harding, Adam J Pawson, Christopher Southan, Jamie A. Davies, Maria P. Abbracchio, Wayne Alexander, Khaled Alhosaini, Magnus Bäck, Nicholas M. Barnes, Ross A. D. Bathgate, Jean‐Martin Beaulieu, Kenneth E. Bernstein, Bernhard Bettler, N.J.M. Birdsall, Victoria A. Blaho, François Boulay, Corinne Bousquet, Hans Bräuner‐Osborne, Geoffrey Burnstock, Girolamo Calò, Justo P. Castaño, Kevin Catt, Stefania Ceruti, Paul L. Chazot, Nan Chiang, Bice Chini, Jerold Chun, Antonia Cianciulli, Olivier Civelli, Lucie H. Clapp, Réjean Couture, Zsolt Csaba, Cláes Dahlgren, Gordon Dent, Khuraijam Dhanachandra Singh, Steven D. Douglas, Pascal Dournaud, Satoru Eguchi, Emanuel Escher, Edward J. Filardo, Tung M. Fong, Marta Fumagalli, Raul R. Gainetdinov, Marc de Gasparo, Craig Gerard, Marvin C. Gershengorn, Fernand Gobeil, Theodore L. Goodfriend, Cyril Goudet, Karen J. Gregory, Andrew L. Gundlach, Jörg Hamann, Julien Hanson, Richard L. Hauger, Debbie L. Hay, Ákos Heinemann, Morley D. Hollenberg, Nicholas D. Holliday, Mastgugu Horiuchi, Daniël Hoyer, László Hunyady, Ahsan Husain, Adriaan P. IJzerman, Tadashi Inagami, Kenneth A. Jacobson, Robert T. Jensen, Ralf Jockers, Deepa Jonnalagadda, Sadashiva S. Karnik, Klemens Kaupmann, Jacqueline Kemp, Charles Kennedy, Yasuyuki Kihara, Takio Kitazawa, Paweł Kozielewicz, Hans‐Jürgen Kreienkamp, Jyrki P. Kukkonen, Tobias Langenhan, Katie Leach, Davide Lecca, John D. Lee, Susan E. Leeman, Jérôme Leprince, Xaria X. Li, Tom A. Williams, Stephen J. Lolait, Amelie Lupp, Robyn Macrae, Janet J. Maguire, Jean Mazella, Craig A. McArdle and 55 more - British Journal of Pharmacology 2021 cited by 488
- International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and Classification of Adenosine Receptors—An Update
Authors: Bertil B. Fredholm, Adriaan P. IJzerman, Kenneth A. Jacobson, Joel Linden, Christa E. Müller - Pharmacological Reviews 2011 cited by 1,291
- Adenosine receptors as therapeutic targets
Authors: Kenneth A. Jacobson, Zhan‐Guo Gao - Nature Reviews Drug Discovery 2006 cited by 1,414
- International Union of Basic and Clinical Pharmacology. CXII: Adenosine Receptors: A Further Update
Authors: Adriaan P. IJzerman, Kenneth A. Jacobson, Christa E. Müller, Bruce N. Cronstein, Rodrigo A. Cunha - Pharmacological Reviews 2022 cited by 152
- Anionic phospholipids control mechanisms of GPCR-G protein recognition
Authors: Naveen Thakur, Arka Prabha Ray, Liam Sharp, Beining Jin, Alexander Duong, Niloofar Gopal Pour, Samuel Obeng, Anuradha V. Wijesekara, Zhan‐Guo Gao, Christopher R. McCurdy, Kenneth A. Jacobson, Edward Lyman, Matthew T. Eddy - Nature Communications 2023 cited by 98
- Two disparate ligand-binding sites in the human P2Y1 receptor
Authors: Dandan Zhang, Zhan‐Guo Gao, Kaihua Zhang, Evgeny Kiselev, Steven Crane, Jiang Wang, Silvia Paoletta, Cuiying Yi, Limin Ma, Wenru Zhang, Gye Won Han, Hong Liu, Vadim Cherezov, Vsevolod Katritch, Hualiang Jiang, Raymond C. Stevens, Kenneth A. Jacobson, Qiang Zhao, Beili Wu - Nature 2015 cited by 370
- Update of P2Y receptor pharmacology: IUPHAR Review 27
Authors: Kenneth A. Jacobson, Esmerilda G. Delicado, Christian Gachet, Charles Kennedy, Ivar von Kügelgen, Beibei Li, María Teresa Miras‐Portugal, Ivana Novak, Torsten Schöneberg, Raquel Pérez‐Sen, Doreen Thor, Beili Wu, Zhenlin Yang, Christa E. Müller - British Journal of Pharmacology 2020 cited by 236
- International Union of Pharmacology LVIII: Update on the P2Y G Protein-Coupled Nucleotide Receptors: From Molecular Mechanisms and Pathophysiology to Therapy
Authors: Maria P. Abbracchio, Geoffrey Burnstock, Jean‐Marie Boeynaems, Eric A. Barnard, José L. Boyer, Charles Kennedy, Gillian E. Knight, Marta Fumagalli, Christian Gachet, Kenneth A. Jacobson, Gary A. Weisman - Pharmacological Reviews 2006 cited by 1,267
- International Union of Pharmacology. XXV. Nomenclature and Classification of Adenosine Receptors
Authors: Bertil B. Fredholm, Adriaan P. IJzerman, Kenneth A. Jacobson, Karl‐Norbert Klotz, Joel Linden - Pharmacological Reviews 2001 cited by 2,558
- Increased Signaling via Adenosine A1 Receptors, Sleep Deprivation, Imipramine, and Ketamine Inhibit Depressive-like Behavior via Induction of Homer1a
Authors: Tsvetan Serchov, Hans‐Willi Clement, Martin K. Schwarz, Felice Iasevoli, Dilip K. Tosh, Marco Idzko, Kenneth A. Jacobson, Andrea de Bartolomeis, Claus Normann, Knut Biber, Dietrich van Calker - Neuron 2015 cited by 211
- Deficiency of adenosine deaminase 2 triggers adenosine-mediated NETosis and TNF production in patients with DADA2
Authors: Carmelo Carmona‐Rivera, Sami S. Khaznadar, Kyawt Shwin, Jorge A. Irizarry‐Caro, Liam J. O’Neil, Yudong Liu, Kenneth A. Jacobson, Amanda K. Ombrello, Deborah L. Stone, Wanxia Li Tsai, Daniel L. Kastner, Ivona Aksentijevich, Mariana J. Kaplan, Peter C. Grayson - Blood 2019 cited by 159
- Structure of the human P2Y12 receptor in complex with an antithrombotic drug
Authors: Kaihua Zhang, Jin Zhang, Zhan‐Guo Gao, Dandan Zhang, Lan Zhu, Gye Won Han, Steven M. Moss, Silvia Paoletta, Evgeny Kiselev, Jane W. Z. Lu, Gustavo Fenalti, Wenru Zhang, Christa E. Müller, Huaiyu Yang, Hualiang Jiang, Vadim Cherezov, Vsevolod Katritch, Kenneth A. Jacobson, Raymond C. Stevens, Beili Wu, Qiang Zhao - Nature 2014 cited by 397
- Allosteric Coupling of Drug Binding and Intracellular Signaling in the A2A Adenosine Receptor
Authors: Matthew T. Eddy, Ming-Yue Lee, Zhan‐Guo Gao, Kate L. White, Tatiana Didenko, Reto Horst, Martin Audet, Paweł Stańczak, Kyle M. McClary, Gye Won Han, Kenneth A. Jacobson, Raymond C. Stevens, Kurt Wüthrich - Cell 2017 cited by 217
- A2A Adenosine Receptor Antagonists in Neurodegenerative Diseases
Authors: Stefania Merighi, Pier Andrea Borea, Katia Varani, Fabrizio Vincenzi, Kenneth A. Jacobson, Stefania Gessi - Current Medicinal Chemistry 2021 cited by 39
- Recent developments in adenosine receptor ligands and their potential as novel drugs
Authors: Christa E. Müller, Kenneth A. Jacobson - Biochimica et Biophysica Acta (BBA) - Biomembranes 2010 cited by 433
- Structural Connection between Activation Microswitch and Allosteric Sodium Site in GPCR Signaling
Authors: Kate L. White, Matthew T. Eddy, Zhan‐Guo Gao, Gye Won Han, Tiffany Lian, Alexander Deary, Nilkanth Patel, Kenneth A. Jacobson, Vsevolod Katritch, Raymond C. Stevens - Structure 2018 cited by 181
- A3Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy
Authors: Kenneth A. Jacobson, Stefania Merighi, Katia Varani, Pier Andrea Borea, Stefania Baraldi, Mojgan Aghazadeh Tabrizi, Romeo Romagnoli, Pier Giovanni Baraldi, Antonella Ciancetta, Dilip K. Tosh, Zhan‐Guo Gao, Stefania Gessi - Medicinal Research Reviews 2017 cited by 152
- A Role for Lipid Shells in Targeting Proteins to Caveolae, Rafts, and Other Lipid Domains
Authors: Richard G.W. Anderson, Kenneth A. Jacobson - Science 2002 cited by 1,118
- Coordinated Adenine Nucleotide Phosphohydrolysis and Nucleoside Signaling in Posthypoxic Endothelium
Authors: Holger K. Eltzschig, Juan C. Ibla, Glenn T. Furuta, Martin O. Leonard, Kenneth A. Jacobson, Keiichi Enjyoji, Simon C. Robson, Sean P. Colgan - The Journal of Experimental Medicine 2003 cited by 495
- Agonist-bound structure of the human P2Y12 receptor
Authors: Jin Zhang, Kaihua Zhang, Zhan‐Guo Gao, Silvia Paoletta, Dandan Zhang, Gye Won Han, Tingting Li, Limin Ma, Wenru Zhang, Christa E. Müller, Huaiyu Yang, Hualiang Jiang, Vadim Cherezov, Vsevolod Katritch, Kenneth A. Jacobson, Raymond C. Stevens, Beili Wu, Qiang Zhao - Nature 2014 cited by 349
