Markus Warmuth
1996–2025 年に発表
- 39
- 論文数
- 18,083
- 被引用数
- 36
- h 指数
- 37
- i10 指数
被引用数
引用元
国・地域
機関
分野
- Biochemistry, Genetics and Molecular Biology51.8%
- Medicine32.4%
- Computer Science9.4%
- Immunology and Microbiology1.8%
- Chemistry1.2%
- Neuroscience0.7%
- その他2.7%
トピック
- Computational Drug Discovery Methods4.4%
- Bioinformatics and Genomic Networks3.3%
- Cancer Genomics and Diagnostics3.2%
- RNA modifications and cancer3%
- Epigenetics and DNA Methylation2.7%
- RNA Research and Splicing2.3%
- その他81.1%
共著者
- Peter Fekkes8
- Silvia Buonamici8
- Nathanael S. Gray6
- Ping Zhu6
- Sung Joon Kim6
- Craig Karr5
- Lihua Yu5
- Michael Hallek5
- Michael Seiler5
- Pavan Kumar5
- William R. Sellers5
- Xiaoling Puyang5
- Alice Loo4
- Crystal MacKenzie4
- Doriano Fabbro4
- Eunice Park4
- Gang Xia4
- Joseph F. Kelleher4
- Laura Corson4
- Marion Dorsch4
- Nicholas Larsen4
- Paul W. Manley4
- Yi Liu4
- Yoshiharu Mizui4
全論文
- The Cancer Cell Line Encyclopedia enables predictive modelling of anticancer drug sensitivity
著者: Jordi Barretina, Giordano Caponigro, Nicolas Stransky, K. Venkatesan, Adam A. Margolin, Sung Joon Kim, Christopher J. Wilson, Joseph Lehár, Gregory V. Kryukov, Dmitriy Sonkin, Anupama Reddy, Manway Liu, Lauren Murray, Michael F. Berger, John E. Monahan, Paula Morais, Jodi Meltzer, Adam Korejwa, Judit Jané‐Valbuena, Felipa Mapa, Joseph Thibault, Eva Bric-Furlong, Pichai Raman, Aaron Shipway, Ingo H. Engels, Jill Cheng, Guoying Karen Yu, Jianjun Yu, Peter Aspesi, Melanie de Silva, Kalpana Jagtap, Michael D. Jones, Li Wang, Charlie Hatton, Emanuele Palescandolo, Supriya Gupta, Scott Mahan, Carrie Sougnez, Robert C. Onofrio, Ted Liefeld, Laura E. MacConaill, Wendy Winckler, Michael Reich, Nanxin Li, Jill P. Mesirov, Stacey Gabriel, Gad Getz, Kristin Ardlie, Vivien W. Chan, Vic E. Myer, Barbara L. Weber, Jeff Porter, Markus Warmuth, Peter M. Finan, Jennifer L. Harris, Matthew Meyerson, Todd R. Golub, Michael Morrissey, William R. Sellers, Robert Schlegel, Levi A. Garraway - Nature 2012 被引用: 8,599
- Allosteric inhibition of SHP2 phosphatase inhibits cancers driven by receptor tyrosine kinases
著者: Ying-Nan P. Chen, Matthew J. LaMarche, Ho Man Chan, Peter Fekkes, Jorge García‐Fortanet, Michael Acker, Brandon Antonakos, Christine Hiu-Tung Chen, Zhouliang Chen, Vesselina G. Cooke, Jason R. Dobson, Zhan Deng, Fei Feng, Brant Firestone, Michelle Fodor, Cary Fridrich, Hui Gao, Denise C. Grünenfelder, Huai-Xiang Hao, Jaison Jacob, Samuel B. Ho, Kathy Hsiao, Kang Zhao, Rajesh Karki, Mitsunori Kato, Jay F. Larrow, Laura R. La Bonte, François Lenoir, Gang Liu, Shumei Liu, Dyuti Majumdar, Matthew J. Meyer, Mark Palermo, Lawrence Perez, Minying Pu, Edmund V. Price, Christopher Quinn, Subarna Shakya, Michael D. Shultz, Joanna Slisz, K. Venkatesan, Ping Wang, Markus Warmuth, Sarah Williams, Guizhi Yang, Jing Yuan, Ji-Hu Zhang, Ping Zhu, Timothy M. Ramsey, Nicholas Keen, William R. Sellers, Travis Stams, Pascal D. Fortin - Nature 2016 被引用: 946
- Discovery of Asciminib (ABL001), an Allosteric Inhibitor of the Tyrosine Kinase Activity of BCR-ABL1
著者: Joseph Schoepfer, Wolfgang Jahnke, Giuliano Berellini, Silvia Buonamici, Simona Cotesta, Sandra W. Cowan‐Jacob, Stephanie Dodd, Peter Drueckes, Doriano Fabbro, Tobias Gabriel, Jean‐Marc Groell, Robert M. Grotzfeld, Amr Hassan, Chrystèle Henry, Varsha Iyer, Darryl Jones, Franco Lombardo, Alice Loo, Paul W. Manley, Xavier Pellé, Gabriele Rummel, Bahaâ Salem, Markus Warmuth, Andrew A. Wylie, Thomas Zöller, Andreas L. Marzinzik, Pascal Furet - Journal of Medicinal Chemistry 2018 被引用: 447
- The allosteric inhibitor ABL001 enables dual targeting of BCR–ABL1
著者: Andrew A. Wylie, Joseph Schoepfer, Wolfgang Jahnke, Sandra W. Cowan‐Jacob, Alice Loo, Pascal Furet, Andreas L. Marzinzik, Xavier Pellé, Jerry Donovan, Wenjing Zhu, Silvia Buonamici, Amr Hassan, Franco Lombardo, Varsha Iyer, Michael R. Palmer, Giuliano Berellini, Stephanie Dodd, Sanjeev Thohan, Hans Bitter, Susan Branford, David M. Ross, Timothy P. Hughes, Lilli Petruzzelli, K. Gary J. Vanasse, Markus Warmuth, Francesco Hofmann, Nicholas Keen, William R. Sellers - Nature 2017 被引用: 614
- H3B-8800, an orally available small-molecule splicing modulator, induces lethality in spliceosome-mutant cancers
著者: Michael Seiler, Akihide Yoshimi, Rachel Darman, Betty Chan, Gregg F. Keaney, Michaël Thomas, Anant A. Agrawal, Benjamin Caleb, Alfredo Csibi, E. Egan Sean, Peter Fekkes, Craig Karr, Virginia M. Klimek, George Lai, Linda Lee, Pavan Kumar, Stanley Chun-Wei Lee, Xiang Liu, Crystal MacKenzie, Carol Meeske, Yoshiharu Mizui, Eric Padron, Eunice Park, Ermira Pazolli, Shouyong Peng, Sudeep Prajapati, Justin Taylor, Teng Teng, John Wang, Markus Warmuth, Huilan Yao, Lihua Yu, Ping Zhu, Omar Abdel‐Wahab, Peter G. Smith, Silvia Buonamici - Nature Medicine 2018 被引用: 510
- Cancer-Associated SF3B1 Hotspot Mutations Induce Cryptic 3′ Splice Site Selection through Use of a Different Branch Point
著者: Rachel Darman, Michael Seiler, Anant A. Agrawal, Kian‐Huat Lim, Shouyong Peng, Daniel Aird, Suzanna Bailey, Erica B. Bhavsar, Betty Chan, Simona Colla, Laura Corson, Jacob Feala, Peter Fekkes, Kana Ichikawa, Gregg F. Keaney, Linda Lee, Pavan Kumar, Kaiko Kunii, Crystal MacKenzie, Mark Matijevic, Yoshiharu Mizui, Khin Than Myint, Eun Sun Park, Xiaoling Puyang, Anand Selvaraj, Michael P. Thomas, Jennifer Tsai, John Y. Wang, Markus Warmuth, Hui Yang, Ping Zhu, Guillermo Garcia‐Manero, Richard R. Furman, Lihua Yu, Peter G. Smith, Silvia Buonamici - Cell Reports 2015 被引用: 463
- Targeting Bcr–Abl by combining allosteric with ATP-binding-site inhibitors
著者: Jianming Zhang, Francisco Adrián, Wolfgang Jahnke, Sandra W. Cowan‐Jacob, Allen G. Li, Roxana E. Iacob, Taebo Sim, John T. Powers, Christine Dierks, Fangxian Sun, Gui-Rong Guo, Qiang Ding, Okram Barun, Yongmun Choi, Amy Wojciechowski, Xianming Deng, Guoxun Liu, Gabriele Fendrich, André Strauss, Navratna Vajpai, Stephan Grzesiek, Tove Tuntland, Yi Liu, Badry Bursulaya, Mohammad Azam, Paul W. Manley, John R. Engen, George Q. Daley, Markus Warmuth, Nathanael S. Gray - Nature 2010 被引用: 606
- H3B-6527 Is a Potent and Selective Inhibitor of FGFR4 in FGF19-Driven Hepatocellular Carcinoma
著者: Jaya Julie Joshi, Heather Coffey, Erik Corcoran, Jennifer J. Tsai, Chia‐Ling Huang, Kana Ichikawa, Sudeep Prajapati, Ming‐Hong Hao, Suzanna Bailey, Jeremy Wu, Victoria Rimkunas, Craig Karr, Vanitha Subramanian, Pavan Kumar, Crystal MacKenzie, Raelene Hurley, Takashi Satoh, Kun Yu, Eunice Park, Nathalie Rioux, Amy Kim, Weidong G. Lai, Lihua Yu, Ping Zhu, Silvia Buonamici, Nicholas Larsen, Peter Fekkes, John Wang, Markus Warmuth, Dominic J. Reynolds, Peter G. Smith, Anand Selvaraj - Cancer Research 2017 被引用: 151
- Loss of function JAK1 mutations occur at high frequency in cancers with microsatellite instability and are suggestive of immune evasion
著者: Lee A. Albacker, Jeremy Wu, Peter Smith, Markus Warmuth, Philip J. Stephens, Ping Zhu, Lihua Yu, Juliann Chmielecki - PLoS ONE 2017 被引用: 137
- Mining the CRBN target space redefines rules for molecular glue–induced neosubstrate recognition
著者: Georg Petzold, Pablo Gaínza, Stefano Annunziato, Ilaria Lamberto, Peter Trenh, Laura A. McAllister, Bradley DeMarco, Laura Schwander, R.D. Bunker, Mary Zlotosch, Rohitha Sriramaratnam, Samuel Gilberto, Gerasimos Langousis, Etienne J. Donckèle, Cynthia Quan, Vaïk Strande, Gian Marco De Donatis, Shanique Alabi, Jessica Alers, Michelle Matysik, Camille Staehly, Aurélie Dubois, Arnaud Osmont, Mackenzie Garskovas, David Lyon, L. Wiedmer, Vladimiras Oleinikovas, Raphael Lieberherr, Nooreen Rubin, Daniel T. Lam, Xavier Lucas, Elisa Liardo, Nina Ilic Widlund, Andreas Ritzén, Ramon Miguel Caceres, Dominico Vigil, Jennifer Tsai, Owen B. Wallace, Marisa Peluso, Amine Sadok, Ralph Tiedt, Alison M. Paterson, Vladislav Zarayskiy, Bernhard Fasching, Débora Bonenfant, Markus Warmuth, John C. Castle, Sharon A. Townson - Science 2025 被引用: 71
- Evasion of immunosurveillance by genomic alterations of PPARγ/RXRα in bladder cancer
著者: Manav Korpal, Xiaoling Puyang, Zhenhua J. Wu, Roland Seiler, Craig Furman, Htoo Zarni Oo, Michael Seiler, Sean Irwin, Vanitha Subramanian, Jaya Julie Joshi, Chris Kedong Wang, Victoria Rimkunas, Davide Tortora, Hua Yang, Namita Kumar, Galina Kuznetsov, Mark Matijevic, Jesse C. Chow, Pavan Kumar, Jian Zou, Jacob Feala, Laura Corson, Ryan E. Henry, Anand Selvaraj, Allison Davis, Kristjan Bloudoff, James J. Douglas, Bernhard Kiss, Morgan E. Roberts, Ladan Fazli, Peter C. Black, Peter Fekkes, Peter G. Smith, Markus Warmuth, Lihua Yu, Ming‐Hong Hao, Nicholas Larsen, Mads Daugaard, Ping Zhu - Nature Communications 2017 被引用: 145
- Interfering with Resistance to Smoothened Antagonists by Inhibition of the PI3K Pathway in Medulloblastoma
著者: Silvia Buonamici, Juliet Williams, Michael Morrissey, Anlai Wang, Ribo Guo, Anthony Vattay, Kathy Hsiao, Jing Yuan, John Green, Beatriz Muñoz, Qunyan Yu, Lance Ostrom, Paul Fordjour, Dustin L. Anderson, John E. Monahan, Joseph F. Kelleher, Stefan Peukert, Shifeng Pan, Xu Wu, Sauveur-Michel Maira, Carlos Garcı́a-Echeverrı́a, Kimberly J. Briggs, D. Neil Watkins, Yung-Mae Yao, Christoph Lengauer, Markus Warmuth, William R. Sellers, Marion Dorsch - Science Translational Medicine 2010 被引用: 554
- Splicing modulators act at the branch point adenosine binding pocket defined by the PHF5A–SF3b complex
著者: Teng Teng, Jennifer Tsai, Xiaoling Puyang, Michael Seiler, Shouyong Peng, Sudeep Prajapati, Daniel Aird, Silvia Buonamici, Benjamin Caleb, Betty Chan, Laura Corson, Jacob Feala, Peter Fekkes, Baudouin Gerard, Craig Karr, Manav Korpal, Xiang Liu, Jason T. Lowe, Yoshiharu Mizui, James Palacino, Eunice Park, Peter G. Smith, Vanitha Subramanian, Zhenhua J. Wu, Jian Zou, Lihua Yu, Agustin Chicas, Markus Warmuth, Nicholas Larsen, Ping Zhu - Nature Communications 2017 被引用: 149
- Synthesis, Structure–Activity Relationships, and in Vivo Efficacy of the Novel Potent and Selective Anaplastic Lymphoma Kinase (ALK) Inhibitor 5-Chloro-N2-(2-isopropoxy-5-methyl-4-(piperidin-4-yl)phenyl)-N4-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine (LDK378) Currently in Phase 1 and Phase 2 Clinical Trials
著者: Thomas H. Marsilje, Wei Pei, Bei Chen, Wenshuo Lu, Tetsuo Uno, Yunho Jin, Tao Jiang, Sung Joon Kim, Nanxin Li, Markus Warmuth, Yelena Sarkisova, Frank F. Sun, Auzon Steffy, AnneMarie Culazzo Pferdekamper, Allen G. Li, Sean B. Joseph, Young Ho Kim, Bo Liu, Tove Tuntland, Xiaoming Cui, Nathanael S. Gray, Ruo W. Steensma, Yongqin Wan, Jiqing Jiang, Greg Chopiuk, Jie Li, W. Perry Gordon, Wendy Richmond, Kevin C. Johnson, Jonathan Chang, Todd Groessl, You-Qun He, Andrew Phimister, J. Alex Aycinena, Christian C. Lee, Badry Bursulaya, Donald S. Karanewsky, H. Martin Seidel, Jennifer L. Harris, Pierre‐Yves Michellys - Journal of Medicinal Chemistry 2013 被引用: 412
- Identification of NVP-TAE684, a potent, selective, and efficacious inhibitor of NPM-ALK
著者: Anna Galkin, Jonathan S. Melnick, Sung Joon Kim, Tami Hood, Nanxin Li, Lintong Li, Gang Xia, Ruo W. Steensma, Greg Chopiuk, Jiqing Jiang, Yongqin Wan, Peter Ding, Yi Liu, Fangxian Sun, Peter G. Schultz, Nathanael S. Gray, Markus Warmuth - National Academy of Sciences, Proceedings of the National Academy of Sciences 2006 被引用: 377
- Discovery of NVP-LDE225, a Potent and Selective Smoothened Antagonist
著者: Shifeng Pan, Xu Wu, Jiqing Jiang, Wenqi Gao, Yongqin Wan, Cheng Dai, Dong Han, Jun Liu, Nathan Englund, Yan Wang, Stefan Peukert, Karen Miller‐Moslin, Jing Yuan, Ribo Guo, Melissa Matsumoto, Anthony Vattay, Yun Jiang, Jeffrey Tsao, Fangxian Sun, AnneMarie Culazzo Pferdekamper, Stephanie Dodd, Tove Tuntland, Wieslawa Maniara, Joseph F. Kelleher, Yung‐Mae Yao, Markus Warmuth, Juliet Williams, Marion Dorsch - ACS Medicinal Chemistry Letters 2010 被引用: 328
- Ba/F3 cells and their use in kinase drug discovery
著者: Markus Warmuth, Sung Joon Kim, Xiang-ju Gu, Gang Xia, Francisco Adrián - Current Opinion in Oncology 2006 被引用: 242
- Discovery of Selective Estrogen Receptor Covalent Antagonists for the Treatment of ERαWT and ERαMUT Breast Cancer
著者: Xiaoling Puyang, Craig Furman, Guo Zhu Zheng, Zhenhua J. Wu, Deepti Banka, Kiran Aithal, Sergei Agoulnik, David M. Bolduc, Silvia Buonamici, Benjamin Caleb, Subhasree Das, Sean Eckley, Peter Fekkes, Ming‐Hong Hao, Andrew Hart, René Houtman, Sean Irwin, Jaya Julie Joshi, Craig Karr, Amy Kim, Namita Kumar, Pavan Kumar, Galina Kuznetsov, Weidong G. Lai, Nicholas Larsen, Crystal MacKenzie, Lesley‐Ann Martin, Diana Melchers, Alyssa Moriarty, Tuong-Vi Nguyen, John D. Norris, Morgan O’Shea, Sunil Pancholi, Sudeep Prajapati, Sujatha Rajagopalan, Dominic J. Reynolds, Victoria Rimkunas, Nathalie Rioux, Ricardo Ribas, Amy Siu, Sasirekha Sivakumar, Vanitha Subramanian, Michaël Thomas, Frédéric H. Vaillancourt, John Wang, Suzanne E. Wardell, Michael J. Wick, Shihua Yao, Lihua Yu, Markus Warmuth, Peter G. Smith, Ping Zhu, Manav Korpal - Cancer Discovery 2018 被引用: 112
- Addendum: The Cancer Cell Line Encyclopedia enables predictive modelling of anticancer drug sensitivity
著者: Jordi Barretina, Giordano Caponigro, Nicolas Stransky, K. Venkatesan, Adam A. Margolin, Sung Joon Kim, Christopher J. Wilson, Joseph Lehár, Gregory V. Kryukov, Dmitriy Sonkin, Anupama Reddy, Manway Liu, Lauren Murray, Michael F. Berger, John E. Monahan, Paula Morais, Jodi Meltzer, Adam Korejwa, Judit Jané‐Valbuena, Felipa Mapa, Joseph Thibault, Eva Bric-Furlong, Pichai Raman, Aaron Shipway, Ingo H. Engels, Jill Cheng, Guoying Karen Yu, Jianjun Yu, Peter Aspesi, Melanie de Silva, Kalpana Jagtap, Michael D. Jones, Li Wang, Charlie Hatton, Emanuele Palescandolo, Supriya Gupta, Scott Mahan, Carrie Sougnez, Robert C. Onofrio, Ted Liefeld, Laura E. MacConaill, Wendy Winckler, Michael Reich, Nanxin Li, Jill P. Mesirov, Stacey Gabriel, Gad Getz, Kristin Ardlie, Vivien W. Chan, Vic E. Myer, Barbara L. Weber, Jeff Porter, Markus Warmuth, Peter M. Finan, Jennifer L. Harris, Matthew Meyerson, Todd R. Golub, Michael Morrissey, William R. Sellers, Robert Schlegel, Levi A. Garraway - Nature 2012 被引用: 112
- Mining the CRBN Target Space Redefines Rules for Molecular Glue-induced Neosubstrate Recognition
著者: Georg Petzold, Pablo Gaínza, Stefano Annunziato, Ilaria Lamberto, Peter Trenh, L. L. McAllister, Bradley DeMarco, Laura Schwander, R.D. Bunker, Mary Zlotosch, Rohitha Sriramaratnam, Samuel Gilberto, Gerasimos Langousis, Etienne J. Donckèle, Chao Quan, Vaïk Strande, Gian Marco De Donatis, Shanique Alabi, Jessica Alers, Michelle Matysik, Camille Staehly, Aurélie Dubois, Arnaud Osmont, Mackenzie Garskovas, David Lyon, L. Wiedmer, Vladimiras Oleinikovas, Raphael Lieberherr, Nooreen Rubin, Daniel T. Lam, Nina Ilic Widlund, Andreas Ritzén, Ramon Miguel Caceres, Dominico Vigil, Jennifer J. Tsai, Owen B. Wallace, Marisa O. Peluso, Amine Sadok, Alison M. Paterson, Vladislav Zarayskiy, Bernhard Fasching, Débora Bonenfant, Markus Warmuth, John Castle, Sharon A. Townson - 2024 被引用: 18
- NAMPT Is the Cellular Target of STF-31-Like Small-Molecule Probes
著者: Drew Adams, Daisuke Ito, Matthew G. Rees, Brinton Seashore‐Ludlow, Xiaoling Puyang, Alex H. Ramos, Jaime H. Cheah, Paul A. Clemons, Markus Warmuth, Ping Zhu, Alykhan F. Shamji, Stuart L. Schreiber - ACS Chemical Biology 2014 被引用: 79
- Expansion of Bcr-Abl-Positive Leukemic Stem Cells Is Dependent on Hedgehog Pathway Activation
著者: Christine Dierks, Ronak Beigi, Gui-Rong Guo, Katja Zirlik, Mario Stegert, Paul W. Manley, Christopher Trussell, Annette Schmitt‐Graeff, Klemens Landwerlin, Hendrik Veelken, Markus Warmuth - Cancer Cell 2008 被引用: 512
- Loss of the tumor suppressor Snf5 leads to aberrant activation of the Hedgehog-Gli pathway
著者: Zainab Jagani, E. Lorena Mora‐Blanco, Courtney G. Sansam, Elizabeth S. McKenna, Boris G. Wilson, Dongshu Chen, Justin Klekota, Pablo Tamayo, Phuong Nguyen, Michael Tolstorukov, Peter J. Park, Yoon-Jae Cho, Kathy Hsiao, Silvia Buonamici, Scott L. Pomeroy, Jill P. Mesirov, Heinz Ruffner, Tewis Bouwmeester, Sarah J. Luchansky, Joshua Murtie, Joseph F. Kelleher, Markus Warmuth, William R. Sellers, Charles W.M. Roberts, Marion Dorsch - Nature Medicine 2010 被引用: 253
- Essential role of stromally induced hedgehog signaling in B-cell malignancies
著者: Christine Dierks, Jovana Grbic, Katja Zirlik, Ronak Beigi, Nathan Englund, Gui-Rong Guo, Hendrik Veelken, Monika Engelhardt, Roland Mertelsmann, Joseph F. Kelleher, Peter G. Schultz, Markus Warmuth - Nature Medicine 2007 被引用: 321
