Philip A. Cole
1972–2025 年に発表
- 別表記
- Philip A Cole
- 154
- 論文数
- 28,346
- 被引用数
- 90
- h 指数
- 147
- i10 指数
被引用数
引用元
国・地域
機関
分野
- Biochemistry, Genetics and Molecular Biology58.1%
- Medicine26.9%
- Neuroscience4.3%
- Immunology and Microbiology3%
- Chemistry2.6%
- Agricultural and Biological Sciences1.9%
- その他3.2%
トピック
- Epigenetics and DNA Methylation7.4%
- Histone Deacetylase Inhibitors Research4.7%
- Genomics and Chromatin Dynamics3.2%
- Protein Degradation and Inhibitors3%
- Cancer-related gene regulation2.9%
- Ubiquitin and proteasome pathways2.7%
- その他76.1%
共著者
- Hanjie Jiang15
- David J. Meyers13
- Kwangwoon Lee12
- Zhipeng A. Wang12
- Jay H. Kalin9
- Nam Chu9
- Samuel D. Whedon9
- Sandra B. Gabelli9
- Jeffrey C. Culhane8
- Rhoda M. Alani8
- Ronen Marmorstein8
- Zan Chen8
- Eunju Nam7
- Beth E. Zucconi6
- Chandrani Mukherjee6
- Mingxuan Wu6
- Wayne W. Hancock6
- Yingming Zhao6
- Yousang Hwang6
- Antonieta L. Salguero5
- Brian B. Liau5
- Daniel R. Dempsey5
- Erin M. Bowers5
- John W. R. Schwabe5
全論文
- Histone Demethylation Mediated by the Nuclear Amine Oxidase Homolog LSD1
著者: Yujiang Geno Shi, Yujiang Geno Shi, Fei Lan, Caitlin Matson, Peter Mulligan, Johnathan R. Whetstine, Philip A. Cole, Robert A. Casero, Yang Shi, Yang Shi - Cell 2004 被引用: 3,996
- Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours
著者: Loren Lasko, Clarissa G. Jakob, Rohinton Edalji, Wei Qiu, Debra Montgomery, Enrico L. DiGiammarino, T. Matt Hansen, Roberto M. Risi, Robin R. Frey, Vlasios Manaves, Bailin Shaw, Mikkel A. Algire, Paul Hessler, Lloyd T. Lam, Tamar Uziel, Emily J. Faivre, Debra C. Ferguson, Fritz G. Buchanan, Ruth L. Martin, Maricel Torrent, Gary G. Chiang, Kannan R. Karukurichi, J. William Langston, Brian T. Weinert, Chunaram Choudhary, Peter de Vries, Arthur F. Kluge, Michael A. Patane, John H. Van Drie, Ce Wang, David McElligott, Ed Kesicki, Ronen Marmorstein, Chaohong Sun, Philip A. Cole, Saul H. Rosenberg, Michael R. Michaelides, Albert Lai, Kenneth D. Bromberg - Nature 2017 被引用: 879
- Time-Resolved Analysis Reveals Rapid Dynamics and Broad Scope of the CBP/p300 Acetylome
著者: Brian T. Weinert, Takeo Narita, Shankha Satpathy, Balaji Srinivasan, Bogi Karbech Hansen, Christian Schölz, William B. Hamilton, Beth E. Zucconi, Wei Wang, Wenshe Ray Liu, Joshua M. Brickman, Edward A. Kesicki, Albert Lai, Kenneth D. Bromberg, Philip A. Cole, Chunaram Choudhary - Cell 2018 被引用: 554
- Protein Lysine Acetylation by p300/CBP
著者: Beverley M. Dancy, Philip A. Cole - Chemical Reviews 2015 被引用: 629
- Ghrelin
著者: Timo D. Müller, Rubén Nogueiras, Mark L. Andermann, Zane B. Andrews, Stefan D. Anker, Jesús Argente, Rachel L. Batterham, S.C. Benoit, C. Y. Bowers, Fabio Broglio, Felipe F. Casanueva, David A. D’Alessio, Inge Depoortere, Allan Geliebter, Ezio Ghigo, Philip A. Cole, Michael A. Cowley, D. E. Cummings, Alain Dagher, Sabrina Diano, Suzanne L. Dickson, Carlos Diéguez, Riccarda Granata, Harvey J. Grill, Kelly Grove, Kirk M. Habegger, Kristy M. Heppner, Mark L. Heiman, Laura M. Holsen, Birgitte Holst, Akio Inui, J-O Jansson, Henriette Kirchner, Márta Korbonits, Blandine Laferrère, C.W. LeRoux, Miguel López, Sophie Morin, Michiko Nakazato, Ralf Nass, Diego Pérez–Tilve, Paul T. Pfluger, Thue W. Schwartz, Randy J. Seeley, Mark W. Sleeman, Yuxiang Sun, Lori Sussel, Jenny Tong, Michael O. Thorner, A. J. van der Lely, L. H. T. Van der Ploeg, Jeffrey M. Zigman, Masayasu Kojima, Kenji Kangawa, R G Smith, Tamás L. Horváth, M. Tschöp - Molecular Metabolism 2015 被引用: 1,008
- Nuclear GTPSCS functions as a lactyl-CoA synthetase to promote histone lactylation and gliomagenesis
著者: Ruilong Liu, Xuelian Ren, Yae Eun Park, Huixu Feng, Xinlei Sheng, Xiaohan Song, Roya AminiTabrizi, Hardik Shah, Lingting Li, Yu Zhang, Kalil G. Abdullah, Sarah DuBois-Coyne, Hening Lin, Philip A. Cole, Ralph J. DeBerardinis, Samuel K. McBrayer, He Huang, Yingming Zhao - Cell Metabolism 2024 被引用: 160
- An Allosteric Mechanism for Activation of the Kinase Domain of Epidermal Growth Factor Receptor
著者: Xuewu Zhang, Jodi Gureasko, Kui Shen, Philip A. Cole, John Kuriyan - Cell 2006 被引用: 1,666
- Acetylation of Tau Inhibits Its Degradation and Contributes to Tauopathy
著者: Sang-Won Min, Seo-Hyun Cho, Yungui Zhou, Sebastian Schroeder, Vahram Haroutunian, William W. Seeley, Eric J. Huang, Yong Shen, Eliezer Masliah, Chandrani Mukherjee, David J. Meyers, Philip A. Cole, Mélanie Ott, Li Gan - Neuron 2010 被引用: 925
- The regulatory enzymes and protein substrates for the lysine β-hydroxybutyrylation pathway
著者: He Huang, Di Zhang, Yejing Weng, Kyle Delaney, Zhanyun Tang, Cong Yan, Shankang Qi, Chao Peng, Philip A. Cole, Robert G. Roeder, Yingming Zhao - Science Advances 2021 被引用: 219
- The Chemical Biology of Reversible Lysine Post-translational Modifications
著者: Zhipeng A. Wang, Philip A. Cole - Cell chemical biology 2020 被引用: 194
- Virtual Ligand Screening of the p300/CBP Histone Acetyltransferase: Identification of a Selective Small Molecule Inhibitor
著者: Erin M. Bowers, Gai Yan, Chandrani Mukherjee, Andrew Orry, Ling Wang, Marc A. Holbert, Nicholas T. Crump, Catherine A. Hazzalin, Glen Liszczak, Hua Yuan, Cecilia Larocca, S. Adrian Saldanha, Ruben Abagyan, Yan Sun, David J. Meyers, Ronen Marmorstein, Louis C. Mahadevan, Rhoda M. Alani, Philip A. Cole - Chemistry & Biology 2010 被引用: 655
- Expressed protein ligation: A general method for protein engineering
著者: Tom W. Muir, Dolan Sondhi, Philip A. Cole - National Academy of Sciences, Proceedings of the National Academy of Sciences 1998 被引用: 1,182
- Targeting the CoREST complex with dual histone deacetylase and demethylase inhibitors
著者: Jay H. Kalin, Muzhou Wu, Andrea V. Gómez, Yun Song, Jayanta Das, Dawn Hayward, Nkosi Adejola, Mingxuan Wu, Izabela Panova, Hye Jin Chung, Edward Kim, Holly Roberts, Justin M. Roberts, Polina Prusevich, Jeliazko R. Jeliazkov, Shourya S. Roy Burman, Louise Fairall, Charles P. Milano, Abdulkerim Eroglu, Charlotte M. Proby, Albena T. Dinkova‐Kostova, Wayne W. Hancock, Jeffrey J. Gray, James E. Bradner, Sérgio Valente, Antonello Mai, Nicole M. Anders, Michelle A. Rudek, Yong Hu, Byungwoo Ryu, John W. R. Schwabe, Andrea Mattevi, Rhoda M. Alani, Philip A. Cole - Nature Communications 2018 被引用: 233
- Mechanism of Crosstalk between the LSD1 Demethylase and HDAC1 Deacetylase in the CoREST Complex
著者: Yun Song, Lisbeth Dagil, Louise Fairall, Naomi Robertson, Mingxuan Wu, Timothy J. Ragan, Christos G. Savva, Almutasem Saleh, Nobuhiro Morone, Micha B. A. Kunze, Andrew G. Jamieson, Philip A. Cole, D. Flemming Hansen, John W. R. Schwabe - Cell Reports 2020 被引用: 141
- Re-programing Chromatin with a Bifunctional LSD1/HDAC Inhibitor Induces Therapeutic Differentiation in DIPG
著者: Jamie N. Anastas, Barry M. Zee, Jay H. Kalin, Mirhee Kim, Robyn Guo, Sanda Alexandrescu, Andrés Blanco, Stefanie Giera, Shawn Gillespie, Jayanta Das, Muzhou Wu, Sarah E. Nocco, Dennis M. Bonal, Quang‐Dé Nguyen, Mario L. Suvà, B Bernstein, Rhoda M. Alani, Todd R. Golub, Philip A. Cole, Mariella G. Filbin, Yang Shi - Cancer Cell 2019 被引用: 191
- Histone H2B Deacylation Selectivity: Exploring Chromatin’s Dark Matter with an Engineered Sortase
著者: Zhipeng A. Wang, Samuel D. Whedon, Mingxuan Wu, Siyu Wang, Edward A. Brown, Ananya Anmangandla, Liam Regan, Kwangwoon Lee, Jianfeng Du, Jun Young Hong, Louise Fairall, Taylor Kay, Hening Lin, Yingming Zhao, John W. R. Schwabe, Philip A. Cole - Journal of the American Chemical Society 2022 被引用: 62
- Regulation of the p300 HAT domain via a novel activation loop
著者: Paul R Thompson, Dongxia Wang, Ling Wang, Marcella Fulco, Natalia Pediconi, Dianzheng Zhang, Woojin An, Qingyuan Ge, Robert G. Roeder, Jiemin Wong, Massimo Levrero, Vittorio Sartorelli, Robert J. Cotter, Philip A. Cole - Nature Structural & Molecular Biology 2004 被引用: 423
- Genetically encoded biosensors for visualizing live-cell biochemical activity at super-resolution
著者: Gary Mo, Brian Ross, Fabian Hertel, Premashis Manna, Xinxing Yang, Eric C. Greenwald, Chris Booth, Ashlee M. Plummer, Brian Tenner, Zan Chen, Yuxiao Wang, Eileen J. Kennedy, Philip A. Cole, Karen G. Fleming, Amy E. Palmer, Ralph Jimenez, Jie Xiao, Peter Dedecker, Jin Zhang - Nature Methods 2017 被引用: 173
- Akt Kinase Activation Mechanisms Revealed Using Protein Semisynthesis
著者: Nam Chu, Antonieta L. Salguero, Albert Z. Liu, Zan Chen, Daniel R. Dempsey, Scott B. Ficarro, William M. Alexander, Jarrod A. Marto, Yana Li, L. Mario Amzel, Sandra B. Gabelli, Philip A. Cole - Cell 2018 被引用: 155
- The structural determinants of PH domain-mediated regulation of Akt revealed by segmental labeling
著者: Nam Chu, Thibault Viennet, Hwan Bae, Antonieta L. Salguero, Andras Boeszoermenyi, Haribabu Arthanari, Philip A. Cole - eLife 2020 被引用: 73
- Structural Basis of Sirtuin 6-Catalyzed Nucleosome Deacetylation
著者: Zhipeng A. Wang, Jonathan Markert, Samuel D. Whedon, Maheeshi Yapa Abeywardana, Kwangwoon Lee, Hanjie Jiang, Carolay Suarez, Hening Lin, Lucas Farnung, Philip A. Cole - Journal of the American Chemical Society 2023 被引用: 58
- A central role for regulated protein stability in the control of TFE3 and MITF by nutrients
著者: Christopher Nardone, Brad A. Palanski, Daniel C. Scott, Richard T. Timms, Karl W. Barber, Xin Gu, Aoyue Mao, Yumei Leng, Emma V. Watson, Brenda A. Schulman, Philip A. Cole, Stephen J. Elledge - Molecular Cell 2023 被引用: 49
- The structural basis of protein acetylation by the p300/CBP transcriptional coactivator
著者: Xin Liu, Ling Wang, Kehao Zhao, Paul R. Thompson, Yousang Hwang, Ronen Marmorstein, Philip A. Cole - Nature 2008 被引用: 445
- The Leukemogenicity of AML1-ETO Is Dependent on Site-Specific Lysine Acetylation
著者: Lan Wang, Alexander Gural, Xiao‐Jian Sun, Xinyang Zhao, Fabiana Perna, Gang Huang, Megan Hatlen, Ly Vu, Fan Liu, Haiming Xu, Takashi Asai, Hao Xu, Tony DeBlasio, Sílvia Menéndez, Francesca Voza, Yanwen Jiang, Philip A. Cole, Jinsong Zhang, Ari Melnick, Robert G. Roeder, Stephen D. Nimer - Science 2011 被引用: 240
