Stefan Knapp
1983–2025 年に発表
- 318
- 論文数
- 42,287
- 被引用数
- 112
- h 指数
- 301
- i10 指数
被引用数
引用元
国・地域
機関
分野
- Biochemistry, Genetics and Molecular Biology56.9%
- Medicine24.2%
- Computer Science6%
- Chemistry4.1%
- Immunology and Microbiology3%
- Neuroscience1.3%
- その他4.5%
トピック
- Protein Degradation and Inhibitors7.8%
- Ubiquitin and proteasome pathways4.3%
- Computational Drug Discovery Methods3.8%
- Histone Deacetylase Inhibitors Research2.7%
- Multiple Myeloma Research and Treatments2.2%
- Epigenetics and DNA Methylation1.9%
- その他77.3%
共著者
- Susanne Müller65
- A. Chaikuad63
- P. Filippakopoulos42
- Benedict‐Tilman Berger32
- O. Fedorov29
- Andreas Krämer24
- Paul E. Brennan22
- Alex N. Bullock21
- Martin P. Schwalm21
- S. Picaud20
- Jonathan M. Elkins19
- Sebastian Mathea19
- Martin Schröder17
- Ewgenij Proschak16
- Nathanael S. Gray16
- Stefan Laufer16
- Thomas Hanke16
- Daniel Merk15
- Jan Heering15
- Martin Philpott15
- Andreas C. Joerger14
- Oleg Fedorov14
- Deep Chatterjee13
- Lena M. Berger13
全論文
- Selective inhibition of BET bromodomains
著者: P. Filippakopoulos, Jun Qi, S. Picaud, Y. Shen, William Smith, O. Fedorov, Elizabeth M. Morse, T. Keates, Tyler Hickman, I. Felletar, Martin Philpott, Shonagh Munro, Michael R. McKeown, Yuchuan Wang, Amanda L. Christie, Nathan West, Michael J. Cameron, Brian E. Schwartz, Tom D. Heightman, Nicholas La Thangue, Christopher A. French, Olaf Wiest, Andrew L. Kung, Stefan Knapp, James E. Bradner - Nature 2010 被引用: 4,337
- Trends in kinase drug discovery: targets, indications and inhibitor design
著者: Misty M. Attwood, Doriano Fabbro, Aleksandr V. Sokolov, Stefan Knapp, Helgi B. Schiöth - Nature Reviews Drug Discovery 2021 被引用: 780
- Histone Recognition and Large-Scale Structural Analysis of the Human Bromodomain Family
著者: P. Filippakopoulos, S. Picaud, Maria Mangos, Tracy Keates, Jean‐Philippe Lambert, Dalia Baršytė-Lovejoy, I. Felletar, Rudolf Volkmer, Susanne Müller, Tony Pawson, Anne‐Claude Gingras, C.H. Arrowsmith, Stefan Knapp - Cell 2012 被引用: 1,777
- Copper is required for oncogenic BRAF signalling and tumorigenesis
著者: Donita C. Brady, Matthew S. Crowe, Michelle L. Turski, G. Aaron Hobbs, Xiaojie Yao, A. Chaikuad, Stefan Knapp, Kunhong Xiao, Sharon L. Campbell, Dennis J. Thiele, Christopher M. Counter - Nature 2014 被引用: 612
- Targeting bromodomains: epigenetic readers of lysine acetylation
著者: P. Filippakopoulos, Stefan Knapp - Nature Reviews Drug Discovery 2014 被引用: 1,245
- Colorectal Cancer Organoid–Stroma Biobank Allows Subtype-Specific Assessment of Individualized Therapy Responses
著者: Henner F. Farin, Mohammed H. Mosa, Benardina Ndreshkjana, Britta M. Grebbin, Birgit Ritter, Constantin Menche, Kilian B. Kennel, Paul K. Ziegler, Lili Szabó, Julia Bollrath, Dietmar Rieder, Birgitta E. Michels, Alena Kress, Müge Bozlar, Tahmineh Darvishi, Sara Stier, Ivan-Maximilano Kur, Katrin Bankov, Rebecca Kesselring, Stefan Fichtner‐Feigl, Bernhard Brüne, Thorsten Oliver Goetze, Salah‐Eddin Al‐Batran, Christian Brandts, Wolf O. Bechstein, Peter J. Wild, Andreas Weigert, Susanne Müller, Stefan Knapp, Zlatko Trajanoski, Florian R. Greten - Cancer Discovery 2023 被引用: 109
- The promise and peril of chemical probes
著者: C.H. Arrowsmith, James E. Audia, Christopher P. Austin, Jonathan B. Baell, Jonathan P. Bennett, Julian Blagg, C. Bountra, Paul E. Brennan, Peter J. Brown, Mark E. Bunnage, Carolyn Buser‐Doepner, Robert M Campbell, Adrian J. Carter, Philip Cohen, Robert A. Copeland, Ben Cravatt, Jayme L. Dahlin, Dashyant Dhanak, A.M. Edwards, Mathias Frederiksen, Stephen V. Frye, Nathanael S. Gray, Charles E. Grimshaw, David Hepworth, Trevor Howe, K. Huber, Jian Jin, Stefan Knapp, Joanne Kotz, Ryan G. Kruger, Derek Lowe, Mary M. Mader, Brian D. Marsden, Anke Mueller‐Fahrnow, Susanne Müller, Rónán C. O’Hagan, John P. Overington, Dafydd R. Owen, Saul H. Rosenberg, Ruth A. Ross, Bryan L. Roth, Matthieu Schapira, Stuart L. Schreiber, Brian K. Shoichet, M. Sundström, Giulio Superti-Furga, Jack Taunton, Leticia Toledo‐Sherman, Chris Walpole, Michael A. Walters, Timothy M. Willson, Paul Workman, Robert N. Young, William J. Zuercher - Nature Chemical Biology 2015 被引用: 850
- PROTAC-mediated degradation reveals a non-catalytic function of AURORA-A kinase
著者: Bikash Adhikari, Jelena Božilović, Mathias Diebold, Jessica Denise Schwarz, Julia Hofstetter, Martin Schröder, Marek Wanior, Ashwin Narain, Markus Vogt, Nevenka Dudvarski Stanković, Apoorva Baluapuri, Lars Schönemann, Lorenz Eing, Pranjali Bhandare, Bernhard Küster, Andreas Schlösser, Stephanie Heinzlmeir, Christoph Sotriffer, Stefan Knapp, Elmar Wolf - Nature Chemical Biology 2020 被引用: 173
- Exploration of Type II Binding Mode: A Privileged Approach for Kinase Inhibitor Focused Drug Discovery?
著者: Zheng Zhao, Hong Wu, Li Wang, Yi Liu, Stefan Knapp, Qingsong Liu, Nathanael S. Gray - ACS Chemical Biology 2014 被引用: 428
- Accurate calculation of the absolute free energy of binding for drug molecules
著者: Matteo Aldeghi, Alexander Heifetz, Michael J. Bodkin, Stefan Knapp, Philip C. Biggin - Chemical Science 2015 被引用: 398
- Quantitative, Wide-Spectrum Kinase Profiling in Live Cells for Assessing the Effect of Cellular ATP on Target Engagement
著者: James D. Vasta, Cesear Corona, Jennifer Wilkinson, Chad Zimprich, James R. Hartnett, Morgan R. Ingold, Kristopher Zimmerman, Thomas Machleidt, Thomas A. Kirkland, Kristin G. Huwiler, Rachel Friedman Ohana, Michael R. Slater, Paul Otto, Mei Cong, Carrow I. Wells, Benedict‐Tilman Berger, Thomas Hanke, Carina Glas, Ke Ding, David H. Drewry, K. Huber, Timothy M. Willson, Stefan Knapp, Susanne Müller, Poncho Meisenheimer, Frank Fan, Keith V. Wood, Matthew B. Robers - Cell chemical biology 2017 被引用: 293
- Structure of LRRK2 in Parkinson’s disease and model for microtubule interaction
著者: Colin K. Deniston, John Salogiannis, Sebastian Mathea, David Snead, Indrajit Lahiri, Mariusz Matyszewski, Oscar Donosa, Reika Watanabe, Jan Böhning, Andrew K. Shiau, Stefan Knapp, Elizabeth Villa, Samara L. Reck‐Peterson, Andrés E. Leschziner - Nature 2020 被引用: 247
- Tracking the PROTAC degradation pathway in living cells highlights the importance of ternary complex measurement for PROTAC optimization
著者: Martin P. Schwalm, Andreas Krämer, Anja Dölle, Janik Weckesser, Xufen Yu, Jian Jin, Krishna Saxena, Stefan Knapp - Cell chemical biology 2023 被引用: 96
- The Cysteinome of Protein Kinases as a Target in Drug Development
著者: A. Chaikuad, Pierre Koch, Stefan Laufer, Stefan Knapp - Angewandte Chemie International Edition 2017 被引用: 238
- Structural Basis for Cul3 Protein Assembly with the BTB-Kelch Family of E3 Ubiquitin Ligases
著者: Peter Canning, C.D.O. Cooper, T. Krojer, James W. Murray, A.C.W. Pike, A. Chaikuad, Tracy Keates, Chancievan Thangaratnarajah, Viktorija Hojzan, Brian D. Marsden, O. Gileadi, Stefan Knapp, F. von Delft, Alex N. Bullock - Journal of Biological Chemistry 2013 被引用: 294
- CBP30, a selective CBP/p300 bromodomain inhibitor, suppresses human Th17 responses
著者: Ariane Hammitzsch, C. Tallant, O. Fedorov, Alison O’Mahony, Paul E. Brennan, Duncan A. Hay, Fernando O. Martínez, Hussein Al‐Mossawi, Jelle de Wit, Matteo Vecellio, Christopher Wells, B P Wordsworth, Susanne Müller, Stefan Knapp, Paul Bowness - National Academy of Sciences, Proceedings of the National Academy of Sciences 2015 被引用: 256
- Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor
著者: Laetitia J. Martin, Manfred Koegl, Gerd Bader, Xiaoling Cockcroft, O. Fedorov, Dennis Fiegen, Thomas Gerstberger, Marco H. Hofmann, Anja Hohmann, Dirk Kessler, Stefan Knapp, Petr Knesl, Stefan Kornigg, Susanne Müller, Herbert Nar, Catherine Rogers, Klaus Rumpel, Otmar Schaaf, Steffen Steurer, C. Tallant, Christopher R. Vakoc, Markus Zeeb, Andreas Zoephel, Mark Pearson, Guido Boehmelt, Darryl B. McConnell - Journal of Medicinal Chemistry 2016 被引用: 224
- Exploiting vulnerabilities of SWI/SNF chromatin remodelling complexes for cancer therapy
著者: Marek Wanior, Andreas Krämer, Stefan Knapp, Andreas C. Joerger - Oncogene 2021 被引用: 165
- CDK11 regulates pre-mRNA splicing by phosphorylation of SF3B1
著者: Milan Hluchý, Pavla Gajdušková, Igor Ruiz de los Mozos, Michal Rájecký, Michael Kluge, Benedict‐Tilman Berger, Zuzana Slabá, David Potěšil, Elena Weiß, Jernej Ule, Zbyněk Zdráhal, Stefan Knapp, Kamil Paruch, Caroline C. Friedel, Dalibor Blažek - Nature 2022 被引用: 90
- RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain
著者: S. Picaud, Christopher Wells, I. Felletar, Deborah H. Brotherton, Sarah Martin, P. Savitsky, Beatriz Díez-Dacal, Martin Philpott, C. Bountra, Hannah Lingard, O. Fedorov, Susanne Müller, Paul E. Brennan, Stefan Knapp, P. Filippakopoulos - National Academy of Sciences, Proceedings of the National Academy of Sciences 2013 被引用: 481
- The ins and outs of selective kinase inhibitor development
著者: Susanne Müller, A. Chaikuad, Nathanael S. Gray, Stefan Knapp - Nature Chemical Biology 2015 被引用: 287
- Discovery and Optimization of Small-Molecule Ligands for the CBP/p300 Bromodomains
著者: Duncan A. Hay, Oleg Fedorov, Sarah Martin, Dean C. Singleton, C. Tallant, Christopher Wells, S. Picaud, Martin Philpott, Octovia Monteiro, Catherine Rogers, Stuart J. Conway, Timothy P. C. Rooney, Anthony Tumber, Clarence Yapp, P. Filippakopoulos, Mark E. Bunnage, Susanne Müller, Stefan Knapp, Christopher J. Schofield, Paul E. Brennan - Journal of the American Chemical Society 2014 被引用: 285
- Mapping the Endothelial Cell S -Sulfhydrome Highlights the Crucial Role of Integrin Sulfhydration in Vascular Function
著者: Sofia‐Iris Bibli, Jiong Hu, Mario Looso, Andreas Weigert, Corina Rațiu, Janina Wittig, Maria Kyriaki Drekolia, Lukas Tombor, Voahanginirina Randriamboavonjy, Matthias S. Leisegang, Philipp Goymann, Fredy Delgado Lagos, Beate Fißlthaler, Sven Zukunft, Anastasia Kyselova, Alberto Fernando Oliveira Justo, Juliana Heidler, Diamantis I. Tsilimigras, Ralf P. Brandes, Stefanie Dimmeler, Andreas Papapetropoulos, Stefan Knapp, Stefan Offermanns, Ilka Wittig, Stephen L. Nishimura, Fragiska Sigala, Ingrid Fleming - Circulation 2020 被引用: 107
- PROTAC degraders as chemical probes for studying target biology and target validation
著者: Václav Němec, Martin P. Schwalm, Susanne Müller, Stefan Knapp - Chemical Society Reviews 2022 被引用: 83
