Richard A. Lerner
Active 1966–2024
- 177
- Papers
- 41,033
- Citations
- 107
- h-index
- 177
- i10-index
Citations
Citation sources
Countries
Institutions
Fields
- Medicine40.8%
- Biochemistry, Genetics and Molecular Biology35.3%
- Chemistry7.2%
- Immunology and Microbiology5.5%
- Agricultural and Biological Sciences2.8%
- Materials Science1.8%
- Other6.6%
Topics
- Monoclonal and Polyclonal Antibodies Research5.8%
- Chemical Synthesis and Analysis3.4%
- Cannabis and Cannabinoid Research3.2%
- Glycosylation and Glycoproteins Research2.6%
- RNA and protein synthesis mechanisms2.2%
- Advanced biosensing and bioanalysis techniques1.4%
- Other81.4%
Coauthors
- Carlos F. Barbas27
- Kim D. Janda24
- Ian A. Wilson21
- Stephen J. Benkovic13
- Guang Yang12
- Jia Xie12
- Hannah Alexander11
- Richard A. Houghten10
- Thomas M. Shinnick10
- Benjamin List9
- Doron Shabat9
- John A. Tainer9
- Peter Wirsching9
- Paul Wentworth8
- Benjamin F. Cravatt7
- Dale L. Boger7
- Frank J. Dixon7
- J G Sutcliffe7
- Peixiang Ma7
- Elizabeth D. Getzoff6
- Guofu Zhong6
- H. Jane Dyson6
- Hongtao Xu6
- J. Gregor Sutcliffe6
All papers
- Encoded combinatorial chemistry.
Authors: Sydney Brenner, Richard A. Lerner - National Academy of Sciences, Proceedings of the National Academy of Sciences 1992 cited by 1,011
- Molecular characterization of an enzyme that degrades neuromodulatory fatty-acid amides
Authors: Benjamin F. Cravatt, Dan K. Giang, Stephen P. Mayfield, Dale L. Boger, Richard A. Lerner, Norton B. Gilula - Nature 1996 cited by 2,131
- DNA-Encoded Chemical Libraries: A Selection System Based on Endowing Organic Compounds with Amplifiable Information
Authors: Dario Neri, Richard A. Lerner - Annual Review of Biochemistry 2018 cited by 363
- Proline-Catalyzed Direct Asymmetric Aldol Reactions
Authors: Benjamin List, Richard A. Lerner, Carlos F. Barbas - Journal of the American Chemical Society 2000 cited by 2,833
- Cross-neutralization of influenza A viruses mediated by a single antibody loop
Authors: Damian C. Ekiert, A.K. Kashyap, John Steel, Adam Rubrum, Gira Bhabha, Reza Khayat, Jeong Hyun Lee, Michael Dillon, Ryann E. O’Neil, Aleksandr M. Faynboym, Michael Horowitz, Lawrence Horowitz, Andrew B. Ward, Peter Palese, Richard J. Webby, Richard A. Lerner, Ramesh R. Bhatt, Ian A. Wilson - Nature 2012 cited by 502
- Regulation of NKT cell-mediated immune responses to tumours and liver inflammation by mitochondrial PGAM5-Drp1 signalling
Authors: Young Jun Kang, Bo‐Ram Bang, Kyung Ho Han, Lixin Hong, Eun-Jin Shim, Jianhui Ma, Richard A. Lerner, Motoyuki Otsuka - Nature Communications 2015 cited by 145
- gem‐Difluoromethylene Alkyne‐Enabled Diverse C−H Functionalization and Application to the on‐DNA Synthesis of Difluorinated Isocoumarins
Authors: Hui Gao, Shuang Lin, Shuning Zhang, Weijie Chen, Xiawen Liu, Guang Yang, Richard A. Lerner, Hongtao Xu, Zhi Zhou, Wei Yi - Angewandte Chemie International Edition 2020 cited by 93
- A Chemistry for Incorporation of Selenium into DNA‐Encoded Libraries
Authors: Hongtao Xu, Yuang Gu, Shuning Zhang, Huan Xiong, Fei Ma, Fengping Lu, Qun Ji, Lili Liu, Peixiang Ma, Wei Hou, Guang Yang, Richard A. Lerner - Angewandte Chemie International Edition 2020 cited by 84
- Elevated levels of oxidized cholesterol metabolites in Lewy body disease brains accelerate α-synuclein fibrilization
Authors: Daryl A. Bosco, Douglas M. Fowler, Qinghai Zhang, Jorgé Nieva, Evan T. Powers, Paul Wentworth, Richard A. Lerner, Jeffery W. Kelly - Nature Chemical Biology 2006 cited by 348
- Diversity of Functionally Permissive Sequences in the Receptor-Binding Site of Influenza Hemagglutinin
Authors: Nicholas C. Wu, Jia Xie, Tianqing Zheng, Corwin M. Nycholat, Geramie Grande, James C. Paulson, Richard A. Lerner, Ian A. Wilson - Cell Host & Microbe 2017 cited by 97
- Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications
Authors: Nicholas Favalli, Gabriele Bassi, Christian Pellegrino, Jacopo Millul, Roberto De Luca, Samuele Cazzamalli, Su Yang, Anika Trenner, Nour L. Mozaffari, Renier Myburgh, Mustafa Moroglu, Stuart J. Conway, Alessandro A. Sartori, Markus G. Manz, Richard A. Lerner, Peter K. Vogt, Jörg Scheuermann, Dario Neri - Nature Chemistry 2021 cited by 77
- Functionality‐Independent DNA Encoding of Complex Natural Products
Authors: Peixiang Ma, Hongtao Xu, Jie Li, Fengping Lu, Fei Ma, Shuyue Wang, Huan Xiong, Wei Wang, Damiano Buratto, Francesco Zonta, Nan Wang, Kaiwen Liu, Tian Hua, Zhi‐Jie Liu, Guang Yang, Richard A. Lerner - Angewandte Chemie 2019 cited by 77
- A complex epistatic network limits the mutational reversibility in the influenza hemagglutinin receptor-binding site
Authors: Nicholas C. Wu, Andrew J. Thompson, Jia Xie, Chih-Wei Lin, Corwin M. Nycholat, Xueyong Zhu, Richard A. Lerner, James C. Paulson, Ian A. Wilson - Nature Communications 2018 cited by 87
- Targeted desialylation and cytolysis of tumour cells by fusing a sialidase to a bispecific T-cell engager
Authors: Zhuo Yang, Yingqin Hou, Geramie Grande, Jong Hyun Cho, Chao Wang, Yujie Shi, Jaroslav Žák, Yue Wan, Ke Qin, Dongfang Liu, John R. Teijaro, Richard A. Lerner, Peng Wu - Nature Biomedical Engineering 2024 cited by 36
- Assembly of combinatorial antibody libraries on phage surfaces: the gene III site.
Authors: Carlos F. Barbas, Angray S. Kang, Richard A. Lerner, Stephen J. Benkovic - National Academy of Sciences, Proceedings of the National Academy of Sciences 1991 cited by 1,187
- Studies on the mechanism of general anesthesia
Authors: Mahmud Arif Pavel, Erling N. Petersen, Hao Wang, Richard A. Lerner, Scott B. Hansen - National Academy of Sciences, Proceedings of the National Academy of Sciences 2020 cited by 209
- Autocrine selection of a GLP-1R G-protein biased agonist with potent antidiabetic effects
Authors: Hongkai Zhang, Emmanuel Sturchler, Jiang Zhu, Ainhoa Nieto, Philip A. Cistrone, Jia Xie, Linling He, Kyungmoo Yea, Teresa M. Jones, Rachel E. Turn, Peter S. Di Stefano, Patrick R. Griffin, Philip E. Dawson, Patricia McDonald, Richard A. Lerner - Nature Communications 2015 cited by 146
- Different genetic barriers for resistance to HA stem antibodies in influenza H3 and H1 viruses
Authors: Nicholas C. Wu, Andrew J. Thompson, Juhye Lee, Wen Su, Britni M. Arlian, Jia Xie, Richard A. Lerner, Hui‐Ling Yen, Jesse D. Bloom, Ian A. Wilson - Science 2020 cited by 77
- Antibody 27F3 Broadly Targets Influenza A Group 1 and 2 Hemagglutinins through a Further Variation in VH1-69 Antibody Orientation on the HA Stem
Authors: Shanshan Lang, Jia Xie, Xueyong Zhu, Nicholas C. Wu, Richard A. Lerner, Ian A. Wilson - Cell Reports 2017 cited by 128
- DNA‐Encoded Compound Libraries as Open Source: A Powerful Pathway to New Drugs
Authors: Richard A. Lerner, Sydney Brenner - Angewandte Chemie International Edition 2017 cited by 119
- Selection of Small Molecules that Bind to and Activate the Insulin Receptor from a DNA-Encoded Library of Natural Products
Authors: Jia Xie, Shuyue Wang, Peixiang Ma, Fei Ma, Jie Li, Wei Wang, Fengping Lu, Huan Xiong, Yuang Gu, Shuning Zhang, Hongtao Xu, Guang Yang, Richard A. Lerner - iScience 2020 cited by 51
- Control of the antitumour activity and specificity of CAR T cells via organic adapters covalently tethering the CAR to tumour cells
Authors: А. В. Степанов, Jia Xie, Qiaoqiao Zhu, Zuyuan Shen, Wenji Su, Letian Kuai, Richard Söll, Christoph Rader, Geramie Shaver, Lacey Douthit, Ding Zhang, R. S. Kalinin, Xiang Fu, Yingying Zhao, Tian Qin, Phil S. Baran, Alexander G. Gabibov, David Bushnell, Dario Neri, Roger D. Kornberg, Richard A. Lerner - Nature Biomedical Engineering 2023 cited by 25
- Expression and assembly of a fully active antibody in algae
Authors: Stephen P. Mayfield, Scott Franklin, Richard A. Lerner - National Academy of Sciences, Proceedings of the National Academy of Sciences 2003 cited by 342
- DNA‐Encoded Libraries: Aryl Fluorosulfonates as Versatile Electrophiles Enabling Facile On‐DNA Suzuki, Sonogashira, and Buchwald Reactions
Authors: Hongtao Xu, Fei Ma, Nan Wang, Wei Hou, Huan Xiong, Fengping Lu, Jie Li, Shuyue Wang, Peixiang Ma, Guang Yang, Richard A. Lerner - Advanced Science 2019 cited by 113
