Markus Schirle
1998–2025 年に発表
- 60
- 論文数
- 18,328
- 被引用数
- 48
- h 指数
- 57
- i10 指数
被引用数
引用元
国・地域
機関
分野
- Biochemistry, Genetics and Molecular Biology57.7%
- Medicine20.2%
- Chemistry9.5%
- Immunology and Microbiology6%
- Computer Science1.8%
- Neuroscience1.1%
- その他3.7%
トピック
- Ubiquitin and proteasome pathways6.2%
- Protein Degradation and Inhibitors5.2%
- Bioinformatics and Genomic Networks4.6%
- Advanced Proteomics Techniques and Applications3.4%
- Wnt/β-catenin signaling in development and cancer2.5%
- Peptidase Inhibition and Analysis2.4%
- その他75.7%
共著者
- John A. Tallarico22
- Jeffrey M. McKenna19
- Daniel K. Nomura18
- Scott M. Brittain17
- Dustin Dovala10
- Jessica N. Spradlin10
- Stefan Stevanović10
- Bernhard Küster7
- Jason R. Thomas7
- Lynn M. McGregor7
- Thomas J. Maimone7
- Hans-Georg Rammensee6
- Michael D. Jones6
- Nathaniel J. Henning6
- Carl C. Ward5
- Hansjörg Schild5
- Jason Murphy5
- Lydia Boike5
- Matthew J. Hesse5
- Tewis Bouwmeester5
- Alexander K. Nussbaum4
- Andreas Bauer4
- Craig Mickanin4
- Frederic Sigoillot4
全論文
- Structure of the DDB1–CRBN E3 ubiquitin ligase in complex with thalidomide
著者: Eric S. Fischer, Kerstin Böhm, John R. Lydeard, Haidi Yang, Michael Stadler, Simone Cavadini, Jane Nagel, Fabrizio C. Serluca, Vincent Acker, Gondichatnahalli M. Lingaraju, Ritesh B. Tichkule, Michael Schebesta, William C. Forrester, Markus Schirle, Ulrich Hassiepen, Johannes Ottl, Marc Hild, Rohan E. J. Beckwith, J. Wade Harper, Jeremy L. Jenkins, Nicolas H. Thomä - Nature 2014 被引用: 1,115
- Selective VPS34 inhibitor blocks autophagy and uncovers a role for NCOA4 in ferritin degradation and iron homeostasis in vivo
著者: William E. Dowdle, Beat Nyfeler, Jane Nagel, R.A. Elling, Shanming Liu, Ellen Triantafellow, Suchithra Menon, Zuncai Wang, Ayako Honda, Gwynn Pardee, John Cantwell, Catherine A. Luu, Iván Cornella‐Taracido, Edmund Harrington, Peter Fekkes, Hong Lei, Qing Fang, Mary Ellen Digan, Debra Burdick, Andrew F. Powers, Stephen B. Helliwell, Simon d‘Aquin, Julie Bastien, Henry Wang, Dmitri Wiederschain, Jenny Kuerth, Philip J. Bergman, David J. Schwalb, Jason R. Thomas, Savuth Ugwonali, Fred Harbinski, John A. Tallarico, Christopher J. Wilson, Vic E. Myer, Jeffery A. Porter, Dirksen E. Bussiere, Peter M. Finan, Mark Labow, Xiaohong Mao, Lawrence G. Hamann, Brendan D. Manning, Reginald Valdez, Thomas Nicholson, Markus Schirle, Mark Knapp, Erin P. Keaney, Leon O. Murphy - Nature Cell Biology 2014 被引用: 740
- Tankyrase inhibition stabilizes axin and antagonizes Wnt signalling
著者: Shih-Min A. Huang, Yuji Mishina, Shanming Liu, Atwood K. Cheung, Frank Stegmeier, Gregory A. Michaud, Olga Charlat, Elizabeth L. Wiellette, Yue Zhang, Stephanie Wiessner, Marc Hild, Xiaoying Shi, Christopher J. Wilson, Craig Mickanin, Vic E. Myer, Aleem Fazal, Ronald Tomlinson, Fabrizio C. Serluca, Wenlin Shao, Hong Cheng, Michael D. Shultz, Christina Rau, Markus Schirle, Judith Schlegl, Sonja Ghidelli, Stephen E. Fawell, Chuang Lu, Daniel Curtis, Marc W. Kirschner, Christoph Lengauer, Peter M. Finan, John A. Tallarico, Tewis Bouwmeester, Jeffery A. Porter, Andreas Bauer, Feng Cong - Nature 2009 被引用: 2,099
- Deubiquitinase-targeting chimeras for targeted protein stabilization
著者: Nathaniel J. Henning, Lydia Boike, Jessica N. Spradlin, Carl C. Ward, Gang Liu, Erika Zhang, Bridget P. Belcher, Scott M. Brittain, Matthew J. Hesse, Dustin Dovala, Lynn M. McGregor, Rachel Valdez Misiolek, Lindsey W. Plasschaert, David J. Rowlands, Feng Wang, Andreas O. Frank, Daniel Fuller, Abigail R. Estes, Katelyn L. Randal, Anoohya Panidapu, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Daniel K. Nomura - Nature Chemical Biology 2022 被引用: 321
- Rational Chemical Design of Molecular Glue Degraders
著者: Ethan S. Toriki, James W. Papatzimas, Kaila Nishikawa, Dustin Dovala, Andreas O. Frank, Matthew J. Hesse, Daniela Danková, Jae-Geun Song, Megan Bruce-Smythe, Heidi Struble, F. García, Scott M. Brittain, Andrew C. Kile, Lynn M. McGregor, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Daniel K. Nomura - ACS Central Science 2023 被引用: 183
- Harnessing the anti-cancer natural product nimbolide for targeted protein degradation
著者: Jessica N. Spradlin, Xirui Hu, Carl C. Ward, Scott M. Brittain, Michael D. Jones, Lisha Ou, Milton To, Andrew Proudfoot, Elizabeth Ornelas, Mikias Woldegiorgis, James A. Olzmann, Dirksen E. Bussiere, Jason R. Thomas, John A. Tallarico, Jeffrey M. McKenna, Markus Schirle, Thomas J. Maimone, Daniel K. Nomura - Nature Chemical Biology 2019 被引用: 424
- Covalent Ligand Screening Uncovers a RNF4 E3 Ligase Recruiter for Targeted Protein Degradation Applications
著者: Carl C. Ward, Jordan I. Kleinman, Scott M. Brittain, Patrick S. Lee, Clive Yik‐Sham Chung, Kenneth H. Kim, Yana Petri, Jason R. Thomas, John A. Tallarico, Jeffrey M. McKenna, Markus Schirle, Daniel K. Nomura - ACS Chemical Biology 2019 被引用: 336
- Discovery of a Covalent FEM1B Recruiter for Targeted Protein Degradation Applications
著者: Nathaniel J. Henning, Andrew G. Manford, Jessica N. Spradlin, Scott M. Brittain, Erika Zhang, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Michael Rapé, Daniel K. Nomura - Journal of the American Chemical Society 2022 被引用: 211
- Chemoproteomics-enabled discovery of covalent RNF114-based degraders that mimic natural product function
著者: Mai Luo, Jessica N. Spradlin, Lydia Boike, Bingqi Tong, Scott M. Brittain, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Thomas J. Maimone, Daniel K. Nomura - Cell chemical biology 2021 被引用: 186
- Chemoproteomics-enabled discovery of a covalent molecular glue degrader targeting NF-κB
著者: Elizabeth A. King, Yoo Jin Cho, Nathan S. Hsu, Dustin Dovala, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Daniel K. Nomura - Cell chemical biology 2023 被引用: 99
- DCAF1-based PROTACs with activity against clinically validated targets overcoming intrinsic- and acquired-degrader resistance
著者: Martin Schröder, Martin Renatus, Xiaoyou Liang, Fabian Meili, Thomas Zöller, Sandrine Ferrand, François Gauter, Xiaoyan Li, Frederic Sigoillot, Scott Gleim, Therese‐Marie Stachyra, Jason R. Thomas, Damien Bégué, Maryam Khoshouei, Peggy Lefeuvre, Rita Andraos-Rey, BoYee Chung, Renate Ma, Benika J. Pinch, Andreas Hofmann, Markus Schirle, Niko Schmiedeberg, Patricia Imbach, Delphine Gorses, Keith Calkins, Beatrice Bauer-Probst, Magdalena Maschlej, Matt Niederst, Rob Maher, Martin Hénault, John Alford, Erik Ahrné, Luca Tordella, Greg Hollingworth, Nicolas H. Thomä, Anna Vulpetti, Thomas Radimerski, Philipp Holzer, Seth Carbonneau, Claudio R. Thoma - Nature Communications 2024 被引用: 88
- Discovery of a Functional Covalent Ligand Targeting an Intrinsically Disordered Cysteine within MYC
著者: Lydia Boike, Alexander G. Cioffi, Felix C. Majewski, Jennifer Co, Nathaniel J. Henning, Michael D. Jones, Gang Liu, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Daniel K. Nomura - Cell chemical biology 2020 被引用: 158
- Proteome survey reveals modularity of the yeast cell machinery
著者: Anne‐Claude Gavin, Patrick Aloy, Paola Grandi, Roland Krause, Markus Böesche, Martina Marzioch, Christina Rau, Lars Juhl Jensen, Sonja Bastuck, Birgit Dümpelfeld, Angela Edelmann, Marie-Anne Heurtier, Verena Hoffman, Christian Hoefert, Karin Klein, Manuela Hudak, Anne‐Marie Michon, Malgorzata Schelder, Markus Schirle, Marita Remor, Tatjana Rudi, Sean Hooper, Andreas Bauer, Tewis Bouwmeester, Georg Casari, Gerard Drewes, Gitte Neubauer, Jens M. Rick, Bernhard Küster, Peer Bork, Robert B. Russell, Giulio Superti‐Furga - Nature 2006 被引用: 2,591
- RNF146 is a poly(ADP-ribose)-directed E3 ligase that regulates axin degradation and Wnt signalling
著者: Yue Zhang, Shanming Liu, Craig Mickanin, Feng Yan, Olga Charlat, Gregory A. Michaud, Markus Schirle, Xiaoying Shi, Marc Hild, Andreas Bauer, Vic E. Myer, Peter M. Finan, Jeffery A. Porter, Shih-Min A. Huang, Feng Cong - Nature Cell Biology 2011 被引用: 434
- Manumycin polyketides act as molecular glues between UBR7 and P53
著者: Yosuke Isobe, Mikiko Okumura, Lynn M. McGregor, Scott M. Brittain, Michael D. Jones, Xiaoyou Liang, R. Larry White, William C. Forrester, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Thomas J. Maimone, Daniel K. Nomura - Nature Chemical Biology 2020 被引用: 134
- Activation of human STING by a molecular glue-like compound
著者: Jie Li, Stephen M. Canham, Hua Wu, Martin Hénault, Lihao Chen, Guoxun Liu, Yu Chen, Gary Yu, Howard Miller, Viktor Horn̆ák, Scott M. Brittain, Gregory A. Michaud, Antonin Tutter, Wendy Broom, Mary Ellen Digan, Sarah M. McWhirter, Kelsey E. Sivick, Helen Trinh Pham, Christine Chen, George S. Tria, Jeffery M. McKenna, Markus Schirle, Xiaohong Mao, Thomas B. Nicholson, Yuan Wang, Jeremy L. Jenkins, Rishi K. Jain, John A. Tallarico, Sejal Patel, Lianxing Zheng, Nathan T. Ross, Charles Y. Cho, Xuewu Zhang, Xiao‐chen Bai, Yan Feng - Nature Chemical Biology 2023 被引用: 71
- Bardoxolone conjugation enables targeted protein degradation of BRD4
著者: Bingqi Tong, Mai Luo, Yi Xie, Jessica N. Spradlin, John A. Tallarico, Jeffrey M. McKenna, Markus Schirle, Thomas J. Maimone, Daniel K. Nomura - Scientific Reports 2020 被引用: 139
- Targeted Protein Degradation through E2 Recruitment
著者: Nafsika Forte, Dustin Dovala, Matthew J. Hesse, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Daniel K. Nomura - ACS Chemical Biology 2023 被引用: 55
- Quantitative mass spectrometry in proteomics: a critical review
著者: Marcus Bantscheff, Markus Schirle, Gavain M.A. Sweetman, Jens M. Rick, Bernhard Küster - Analytical and Bioanalytical Chemistry 2007 被引用: 1,661
- A physical and functional map of the human TNF-α/NF-κB signal transduction pathway
著者: Tewis Bouwmeester, Angela Bauch, Heinz Ruffner, Pierre‐Olivier Angrand, Giovanna Bergamini, Karen Croughton, Cristina-Maria Cruciat, Dirk Eberhard, Julien Gagneur, Sonja Ghidelli, Carsten Hopf, Bettina Huhse, Raffaella Mangano, Anne‐Marie Michon, Markus Schirle, Judith Schlegl, Markus S. Schwab, Martin Stein, Andreas Bauer, Georg Casari, Gerard Drewes, Anne‐Claude Gavin, David Jackson, Gérard Joberty, Gitte Neubauer, Jens M. Rick, Bernhard Küster, Giulio Superti‐Furga - Nature Cell Biology 2004 被引用: 1,028
- Dermcidin: a novel human antibiotic peptide secreted by sweat glands
著者: Birgit Schittek, Rainer Hipfel, Birgit Sauer, Jürgen Bauer, Hubert Kalbacher, Stefan Stevanović, Markus Schirle, Kristina Schroeder, Nikolaus Blin, Friedegund Meier, G. Rassner, Claus Garbe - Nature Immunology 2001 被引用: 735
- Natural products reveal cancer cell dependence on oxysterol-binding proteins
著者: Anthony W. G. Burgett, Thomas B. Poulsen, Kittikhun Wangkanont, D. Ryan Anderson, Chikako Kikuchi, Kousei Shimada, Shuichi Okubo, Kevin C. Fortner, Yoshihiro Mimaki, Minpei Kuroda, Jason Murphy, David J. Schwalb, Eugene C. Petrella, Iván Cornella‐Taracido, Markus Schirle, John A. Tallarico, Matthew D. Shair - Nature Chemical Biology 2011 被引用: 261
- A Nimbolide-Based Kinase Degrader Preferentially Degrades Oncogenic BCR-ABL
著者: Bingqi Tong, Jessica N. Spradlin, Luiz F. T. Novaes, Erika Zhang, Xirui Hu, Malte Moeller, Scott M. Brittain, Lynn M. McGregor, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Thomas J. Maimone, Daniel K. Nomura - ACS Chemical Biology 2020 被引用: 110
- Donor–Acceptor Pyridinium Salts for Photo-Induced Electron-Transfer-Driven Modification of Tryptophan in Peptides, Proteins, and Proteomes Using Visible Light
著者: Caleb Hoopes, Francisco J. Garcia, Akash Mamon Sarkar, Nicholas Kuehl, David T. Barkan, Nicole Collins, Glenna E. Meister, Taylor R. Bramhall, Chien-Hsiang Hsu, Michael D. Jones, Markus Schirle, Michael T. Taylor - Journal of the American Chemical Society 2022 被引用: 69
