Gerard Drewes
1992–2024 年に発表
- 72
- 論文数
- 26,679
- 被引用数
- 57
- h 指数
- 72
- i10 指数
被引用数
引用元
国・地域
機関
分野
- Biochemistry, Genetics and Molecular Biology58.4%
- Medicine23.5%
- Immunology and Microbiology5.1%
- Chemistry5.1%
- Computer Science2.6%
- Neuroscience2.2%
- その他3.1%
トピック
- Bioinformatics and Genomic Networks6.1%
- Alzheimer's disease research and treatments4%
- Protein Degradation and Inhibitors3.8%
- Computational Drug Discovery Methods3.4%
- Ubiquitin and proteasome pathways2.5%
- Protein Structure and Dynamics2.4%
- その他77.8%
共著者
- Marcus Bantscheff26
- Eva‐Maria Mandelkow12
- Sonja Ghidelli‐Disse12
- Carsten Hopf11
- Paola Grandi11
- Dirk Eberhard10
- Gérard Joberty10
- Anne‐Marie Michon9
- Thilo Werner9
- Jacek Biernat8
- Markus Böesche8
- Mikhail M. Savitski8
- Chun‐wa Chung7
- Friedrich Reinhard7
- Maria Fälth Savitski7
- Bernhard Küster6
- Eckhard Mandelkow�6
- Gitte Neubauer6
- Rab K. Prinjha6
- Tewis Bouwmeester6
- Antje Dittmann5
- Bernhard Trinczek5
- Andreas Bauer4
- Andreas Ebneth4
全論文
- Tracking cancer drugs in living cells by thermal profiling of the proteome
著者: Mikhail M. Savitski, Mikhail M. Savitski, Friedrich Reinhard, Holger Franken, Thilo Werner, Maria Fälth Savitski, Maria Fälth Savitski, Dirk Eberhard, Daniel Martinez Molina, Rozbeh Jafari, Rebecca Dovega, Susan Klaeger, Bernhard Küster, P. Nordlund, Marcus Bantscheff, Gerard Drewes - Science 2014 被引用: 1,233
- Inhibition of PAD4 activity is sufficient to disrupt mouse and human NET formation
著者: Huw D. Lewis, John Liddle, Jim Coote, Stephen J. Atkinson, Michael D. Barker, B.D. Bax, Kevin L. Bicker, Ryan P. Bingham, Matthew Campbell, Yu Hua Chen, Chun‐wa Chung, Peter D. Craggs, Rob P. Davis, Dirk Eberhard, Gérard Joberty, Kenneth Lind, Kelly Locke, Claire Maller, Kimberly Martinod, Chris Patten, Oxana Polyakova, Cecil Rise, Martin Rüdiger, Robert J. Sheppard, Daniel J. Slade, Pamela J. Thomas, Jim Thorpe, Gang Yao, Gerard Drewes, Denisa D. Wagner, Paul R Thompson, Rab K. Prinjha, David M. Wilson - Nature Chemical Biology 2015 被引用: 760
- Thermal proteome profiling for unbiased identification of direct and indirect drug targets using multiplexed quantitative mass spectrometry
著者: Holger Franken, Toby Mathieson, Dorothee Childs, Gavain M.A. Sweetman, Thilo Werner, Ina Tögel, Carola Doce, Stephan Gade, Marcus Bantscheff, Gerard Drewes, Friedrich Reinhard, Wolfgang Huber, Mikhail M. Savitski - Nature Protocols 2015 被引用: 708
- Inhibition of BET recruitment to chromatin as an effective treatment for MLL-fusion leukaemia
著者: Mark A. Dawson, Rab K. Prinjha, Antje Dittmann, George Giotopoulos, Marcus Bantscheff, Wai-In Chan, Samuel C. Robson, Chun‐wa Chung, Carsten Hopf, Mikhail M. Savitski, Carola Huthmacher, Emma Gudgin, Dave Lugo, Sören Beinke, Trevor Chapman, Emma J. Roberts, Peter E. Soden, Kurt R. Auger, Olivier Mirguet, Konstanze Doehner, Ruud Delwel, Alan K. Burnett, Philip D. Jeffrey, Gerard Drewes, Kevin Lee, Brian J.P. Huntly, Tony Kouzarides - Nature 2011 被引用: 1,532
- Selective targeting of BD1 and BD2 of the BET proteins in cancer and immunoinflammation
著者: Omer Gilan, Inmaculada Rioja, Kathy Knezevic, Matthew Bell, Miriam M. Yeung, Nicola Harker, Enid Y.N. Lam, Chun‐wa Chung, Paul Bamborough, M. Petretich, Marjeta Urh, Stephen J. Atkinson, Anna K. Bassil, Emma J. Roberts, Dane Vassiliadis, Marian L. Burr, Alex Preston, Christopher R. Wellaway, Thilo Werner, James R. Gray, Anne‐Marie Michon, Thomas Gobbetti, Vinod Kumar, Peter E. Soden, Andrea Haynes, Johanna Vappiani, David F. Tough, S. Taylor, Sarah‐Jane Dawson, Marcus Bantscheff, Matthew Lindon, Gerard Drewes, Emmanuel H. Demont, Danette L. Daniels, Paola Grandi, Rab K. Prinjha, Mark A. Dawson - Science 2020 被引用: 428
- A selective jumonji H3K27 demethylase inhibitor modulates the proinflammatory macrophage response
著者: Laurens Kruidenier, Chun‐wa Chung, Zhongjun Cheng, John Liddle, KaHing Che, Gérard Joberty, Marcus Bantscheff, C. Bountra, Angela Bridges, Hawa Diallo, Dirk Eberhard, Sue Hutchinson, Emma J. Jones, Roy Katso, Melanie Leveridge, Palwinder K. Mander, J. Mosley, César Ramírez-Molina, Paul Rowland, Christopher J. Schofield, Robert J. Sheppard, Julia E. Smith, Catherine Swales, Robert D. Tanner, Pamela J. Thomas, Anthony Tumber, Gerard Drewes, Udo Oppermann, Dinshaw J. Patel, Kevin Lee, David M. Wilson - Nature 2012 被引用: 968
- Functional organization of the yeast proteome by systematic analysis of protein complexes
著者: Anne‐Claude Gavin, Markus Bösche, Roland Krause, Paola Grandi, Martina Marzioch, Andreas Bauer, Jörg Schultz, Jens M. Rick, Anne‐Marie Michon, Cristina‐Maria Cruciat, Marita Remor, Christian R. Höfert, Malgorzata Schelder, Miro Brajenovic, Heinz Ruffner, Alejandro Merino, Karin Klein, Manuela Hudak, David Dickson, Tatjana Rudi, Volker Gnau, Angela Bauch, Sonja Bastuck, Bettina Huhse, Christina Leutwein, Marie-Anne Heurtier, Richard R. Copley, Angela Edelmann, Erich Querfurth, Vladimir Rybin, Gerard Drewes, Manfred Raida, Tewis Bouwmeester, Peer Bork, Bertrand Séraphin, Bernhard Küster, Gitte Neubauer, Giulio Superti‐Furga - Nature 2002 被引用: 4,805
- Proteome survey reveals modularity of the yeast cell machinery
著者: Anne‐Claude Gavin, Patrick Aloy, Paola Grandi, Roland Krause, Markus Böesche, Martina Marzioch, Christina Rau, Lars Juhl Jensen, Sonja Bastuck, Birgit Dümpelfeld, Angela Edelmann, Marie-Anne Heurtier, Verena Hoffman, Christian Hoefert, Karin Klein, Manuela Hudak, Anne‐Marie Michon, Malgorzata Schelder, Markus Schirle, Marita Remor, Tatjana Rudi, Sean Hooper, Andreas Bauer, Tewis Bouwmeester, Georg Casari, Gerard Drewes, Gitte Neubauer, Jens M. Rick, Bernhard Küster, Peer Bork, Robert B. Russell, Giulio Superti‐Furga - Nature 2006 被引用: 2,591
- The International Human Epigenome Consortium: A Blueprint for Scientific Collaboration and Discovery
著者: H.G. Stunnenberg, Sergio Abrignani, David J. Adams, Melanie de Almeida, Lucia Altucci, Viren Amin, Ido Amit, Stylianos E. Antonarakis, Samuel Aparício, Takahiro Arima, Laura Arrigoni, Rob J.W. Arts, Vahid Asnafi, Manel Esteller, Jae‐Bum Bae, Kevin Baßler, Stephan Beck, Benjamin E. Berkman, B Bernstein, Mikhail Bilenky, Adrian Bird, Christoph Bock, Bernhard O. Boehm, Guillaume Bourque, Charles E. Breeze, Benedikt Brors, David Bujold, Oliver S. Burren, Marion J.G. Bussemakers, Adam S. Butterworth, Elı́as Campo, Enrique Carrillo de Santa Pau, Lisa H. Chadwick, Kui Ming Chan, Wei Chen, Tom H. Cheung, Luca Chiapperino, Nak Hyen Choi, Ho‐Ryun Chung, Laura Clarke, Joseph M. Connors, Philippe Cronet, John Danesh, Manolis Dermitzakis, Gerard Drewes, Pawel Durek, Stephanie O. M. Dyke, Tomasz Dyląg, Connie J. Eaves, Peter Ebert, Roland Eils, Jürgen Eils, Catherine Ennis, Tariq Enver, Elise A. Feingold, Bärbel Felder, Anne C. Ferguson‐Smith, Jude Fitzgibbon, Paul Flicek, Roger Foo, Peter Fraser, Mattia Frontini, Eileen E. M. Furlong, Sitanshu Gakkhar, Nina Gasparoni, Gilles Gasparoni, Daniel H. Geschwind, Petar Glažar, Thomas Graf, Frank Grosveld, Xin‐Yuan Guan, Roderic Guigó, Marta Gut, Alf Hamann, Bok-Ghee Han, R. Alan Harris, Simon Heath, Kristian Helin, Jan G. Hengstler, Alireza Heravi‐Moussavi, Karl Herrup, Steven Hill, Jason A. Hilton, Benjamin C. Hitz, Bernhard Horsthemke, Ming Hu, Jooyeon Hwang, Nancy Y. Ip, Takashi Ito, Biola M. Javierre, Sasa Jenko, Thomas Jenuwein, Yann Joly, Steven J.M. Jones, Yae Kanai, Hee Gyung Kang, Aly Karsan, Alexandra K. Kiemer, Song Cheol Kim, Bong-Jo Kim ほか 130 名 - Cell 2016 被引用: 566
- Chemoproteomics profiling of HDAC inhibitors reveals selective targeting of HDAC complexes
著者: Marcus Bantscheff, Carsten Hopf, Mikhail M. Savitski, Antje Dittmann, Paola Grandi, Anne‐Marie Michon, Judith Schlegl, Yann Abraham, Isabelle Becher, Giovanna Bergamini, Markus Böesche, Manja Delling, Birgit Dümpelfeld, Dirk Eberhard, Carola Huthmacher, Toby Mathieson, Daniel Poeckel, Valérie Reader, Katja Strunk, Gavain M.A. Sweetman, Ulrich Kruse, Gitte Neubauer, Nigel G. Ramsden, Gerard Drewes - Nature Biotechnology 2011 被引用: 666
- A physical and functional map of the human TNF-α/NF-κB signal transduction pathway
著者: Tewis Bouwmeester, Angela Bauch, Heinz Ruffner, Pierre‐Olivier Angrand, Giovanna Bergamini, Karen Croughton, Cristina-Maria Cruciat, Dirk Eberhard, Julien Gagneur, Sonja Ghidelli, Carsten Hopf, Bettina Huhse, Raffaella Mangano, Anne‐Marie Michon, Markus Schirle, Judith Schlegl, Markus S. Schwab, Martin Stein, Andreas Bauer, Georg Casari, Gerard Drewes, Anne‐Claude Gavin, David Jackson, Gérard Joberty, Gitte Neubauer, Jens M. Rick, Bernhard Küster, Giulio Superti‐Furga - Nature Cell Biology 2004 被引用: 1,028
- Increased expression of BIN1 mediates Alzheimer genetic risk by modulating tau pathology
著者: Julien Chapuis, Franck Hansmannel, Marc Gistelinck, A Mounier, Caroline Van Cauwenberghe, Kristof Van Kolen, Frank Geller, Yoann Sottejeau, Denise Harold, Pierre Dourlen, Benjamin Grenier‐Boley, Y Kamatani, B. Delepine, Florie Demiautte, Diana Zélénika, Nadège Zommer, Malika Hamdane, Céline Bellenguez, Dartigues Jf, J J Hauw, Florent Letronne, A-M Ayral, Kristel Sleegers, Ann Schellens, Lies Vanden Broeck, Sebastiaan Engelborghs, Peter Paul De Deyn, Rik Vandenberghe, Michael O‘Donovan, Michael J. Owen, Jacques Epelbaum, Marc Mercken, Eric Karran, Marcus Bantscheff, Gerard Drewes, Gérard Joberty, Dominique Campion, J-N Octave, Claudine Berr, Mark Lathrop, Patrick Callaerts, David M. A. Mann, Julie Williams, Luc Buée, Ilse Dewachter, Christine Van Broeckhoven, Philippe Amouyel, Dieder Moechars, Bart Dermaut, J-C Lambert - Molecular Psychiatry 2013 被引用: 440
- Phosphorylation of Ser262 strongly reduces binding of tau to microtubules: Distinction between PHF-like immunoreactivity and microtubule binding
著者: Jacek Biernat, N. Gustke, Gerard Drewes, Eva‐Maria Mandelkow, Eckhard Mandelkow� - Neuron 1993 被引用: 791
- Tau interactome mapping based identification of Otub1 as Tau deubiquitinase involved in accumulation of pathological Tau forms in vitro and in vivo
著者: Peng Wang, Gérard Joberty, Arjan Buist, Alexandre Vanoosthuyse, Ilie‐Cosmin Stancu, Bruno Vasconcelos, Nathalie Pierrot, Maria Faelth-Savitski, Pascal Kienlen‐Campard, Jean‐Noël Octave, Marcus Bantscheff, Gerard Drewes, Diederik Moechars, Ilse Dewachter - Acta Neuropathologica 2017 被引用: 117
- MARK, a Novel Family of Protein Kinases That Phosphorylate Microtubule-Associated Proteins and Trigger Microtubule Disruption
著者: Gerard Drewes, Andreas Ebneth, Ute Preuß, Eva‐Maria Mandelkow, Eckhard Mandelkow� - Cell 1997 被引用: 878
- Thermal proteome profiling monitors ligand interactions with cellular membrane proteins
著者: Friedrich Reinhard, Dirk Eberhard, Thilo Werner, Holger Franken, Dorothee Childs, Carola Doce, Maria Fälth Savitski, Wolfgang Huber, Marcus Bantscheff, Mikhail M. Savitski, Gerard Drewes, Mikhail M. Savitski, Gerard Drewes - Nature Methods 2015 被引用: 319
- Biological plasticity rescues target activity in CRISPR knock outs
著者: Arne H. Smits, Frederik Ziebell, Gérard Joberty, Nico Zinn, William F. Mueller, Sandra Clauder‐Münster, Dirk Eberhard, Maria Fälth Savitski, Paola Grandi, Petra Jakob, Anne‐Marie Michon, Han Sun, Karen Tessmer, Tilmann Bürckstümmer, Marcus Bantscheff, Lars M. Steinmetz, Gerard Drewes, Wolfgang Huber - Nature Methods 2019 被引用: 237
- Quantitative chemical proteomics reveals mechanisms of action of clinical ABL kinase inhibitors
著者: Marcus Bantscheff, Dirk Eberhard, Yann Abraham, Sonja Bastuck, Markus Böesche, Scott Hobson, Toby Mathieson, Jessica Perrin, Manfred Raida, Christina Rau, Valérie Reader, Gavain M.A. Sweetman, Andreas Bauer, Tewis Bouwmeester, Carsten Hopf, Ulrich Kruse, Gitte Neubauer, Nigel G. Ramsden, Jens M. Rick, Bernhard Küster, Gerard Drewes - Nature Biotechnology 2007 被引用: 1,044
- Discovery of I-BRD9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition
著者: Natalie H. Theodoulou, Paul Bamborough, Andrew J. Bannister, Isabelle Becher, Rino A. Bit, Ka Hing, Chun‐wa Chung, Antje Dittmann, Gerard Drewes, David H. Drewry, Laurie Gordon, Paola Grandi, Melanie Leveridge, Matthew Lindon, Anne‐Marie Michon, Mária Judit Molnár, Samuel C. Robson, Nicholas C. O. Tomkinson, Tony Kouzarides, Rab K. Prinjha, P. G. Humphreys - Journal of Medicinal Chemistry 2015 被引用: 234
- Microtubule-associated Protein/Microtubule Affinity-regulating Kinase (p110mark)
著者: Helmut E. Meyer, Eva‐Maria Mandelkow, Eva-Maria Mandelkow, Gerard Drewes, Bernhard Trinczek, Susanne Illenberger, Jacek Biernat, Gerold Schmitt‐Ulms, Eckhard Mandelkow, Eckhard Mandelkow - Journal of Biological Chemistry 1995 被引用: 376
- Click chemistry enables preclinical evaluation of targeted epigenetic therapies
著者: Dean Tyler, Johanna Vappiani, Tatiana Cañeque, Enid Y.N. Lam, Aoife Ward, Omer Gilan, Yih-Chih Chan, Antje Hienzsch, Anna Rutkowska, Thilo Werner, Anne J. Wagner, Dave Lugo, Richard Gregory, César Ramírez Molina, Neil Garton, Christopher R. Wellaway, Susan Jackson, Laura MacPherson, Margarida L. A. Figueiredo, Sabine Stolzenburg, Charles C. Bell, Colin M. House, Sarah‐Jane Dawson, Edwin D. Hawkins, Gerard Drewes, Rab K. Prinjha, Raphaël Rodriguez, Paola Grandi, Mark A. Dawson - Science 2017 被引用: 143
- Antimalarial efficacy of MMV390048, an inhibitor of Plasmodium phosphatidylinositol 4-kinase
著者: Tanya Paquet, Claire Le Manach, Diego González Cabrera, Yassir Younis, Philipp P. Henrich, Tara S. Abraham, Lee M, Rajshekhar Basak, Sonja Ghidelli‐Disse, María José Lafuente-Monasterio, Marcus Bantscheff, Andrea Ruecker, Andrew M. Blagborough, Sara E. Zakutansky, Anne‐Marie Zeeman, Karen L. White, David M. Shackleford, Janne Mannila, Julia Morizzi, Christian Scheurer, Íñigo Angulo‐Barturen, Maria Santos Martínez, Santiago Ferrer, Laura M. Sanz, Francisco‐Javier Gamo, Janette Reader, Mariëtte Botha, Koen J. Dechering, Robert W. Sauerwein, Anchalee Tungtaeng, Pattaraporn Vanachayangkul, Chek Shik Lim, Jeremy N. Burrows, Michael J. Witty, Kennan C. Marsh, Christophe Bodenreider, Rosemary Rochford, Suresh Solapure, Marı́a Belén Jiménez-Dı́az, Sergio Wittlin, Susan A. Charman, Cristina Donini, Brice Campo, Lyn‐Marié Birkholtz, Kirsten K. Hanson, Gerard Drewes, Clemens H. M. Kocken, Michael J. Delves, Didier Leroy, David A. Fidock, David Waterson, Leslie J. Street, Kelly Chibale - Science Translational Medicine 2017 被引用: 272
- Cyclin-dependent kinase 12 is a drug target for visceral leishmaniasis
著者: Susan Wyllie, Michael G. Thomas, Stephen Patterson, Sabrinia Crouch, Manu De Rycker, Rhiannon Lowe, Stephanie Gresham, Michael D. Urbaniak, Thomas D. Otto, Laste Stojanovski, Frederick R. C. Simeons, Sujatha Manthri, Lorna MacLean, Fabio Zuccotto, Nadine Homeyer, Hannah Pflaumer, Markus Böesche, Lalitha Sastry, Paul Connolly, Sébastien Albrecht, Matthew Berriman, Gerard Drewes, David W. Gray, Sonja Ghidelli‐Disse, Susan Dixon, José M. Fiandor, Paul G. Wyatt, Michael A. J. Ferguson, Alan H. Fairlamb, Timothy J. Miles, Kevin D. Read, Ian H. Gilbert - Nature 2018 被引用: 145
- The anticancer human mTOR inhibitor sapanisertib potently inhibits multiple Plasmodium kinases and life cycle stages
著者: Lauren B. Arendse, James M. Murithi, Tarrick Qahash, Charisse Flerida A. Pasaje, Luiz C. Godoy, Sumanta Dey, Liezl Gibhard, Sonja Ghidelli‐Disse, Gerard Drewes, Marcus Bantscheff, María José Lafuente-Monasterio, Stephen Fienberg, Lynn Wambua, Samuel Gachuhi, Dina Coertzen, Mariëtte van der Watt, Janette Reader, Ayesha S. Aswat, Erica Erlank, Nelius Venter, Nimisha Mittal, Madeline R. Luth, Sabine Ottilie, Elizabeth A. Winzeler, Lizette L. Koekemoer, Lyn‐Marié Birkholtz, Jacquin C. Niles, Manuel Llinás, David A. Fidock, Kelly Chibale - Science Translational Medicine 2022 被引用: 46
