Bryan L. Roth
1982–2025 年に発表
- 別表記
- Bryan L Roth
- 284
- 論文数
- 68,512
- 被引用数
- 138
- h 指数
- 280
- i10 指数
被引用数
引用元
国・地域
機関
分野
- Biochemistry, Genetics and Molecular Biology29.4%
- Neuroscience25.2%
- Medicine21%
- Computer Science11.6%
- Psychology4.8%
- Immunology and Microbiology2.1%
- その他5.9%
トピック
- Receptor Mechanisms and Signaling6.9%
- Computational Drug Discovery Methods5.6%
- Neuroscience and Neuropharmacology Research4.4%
- Neurotransmitter Receptor Influence on Behavior3.8%
- Neuropeptides and Animal Physiology3.3%
- Tryptophan and brain disorders1.5%
- その他74.5%
共著者
- Xi‐Ping Huang74
- Brian K. Shoichet32
- Jeffrey F. DiBerto28
- Jian Jin26
- B. Krumm24
- John D. McCorvy22
- Tao Che21
- Vincent Setola20
- Vsevolod Katritch20
- Yongfeng Liu20
- Wesley K. Kroeze19
- Reid H. J. Olsen17
- Samuel T. Slocum17
- Ryan H. Gumpper15
- John J. Irwin14
- Jonathan F. Fay13
- Raymond C. Stevens13
- William C. Wetsel13
- Vadim Cherezov12
- Daniel Wacker11
- Shicheng Zhang11
- Can Cao10
- Gye Won Han10
- Kuglae Kim10
全論文
- Relating protein pharmacology by ligand chemistry
著者: Michael J. Keiser, Bryan L. Roth, Blaine N. Armbruster, Paul Ernsberger, John J. Irwin, Brian K. Shoichet - Nature Biotechnology 2007 被引用: 2,400
- DREADDs for Neuroscientists
著者: Bryan L. Roth - Neuron 2016 被引用: 1,793
- Rapid, reversible activation of AgRP neurons drives feeding behavior in mice
著者: Michael J. Krashes, Shuichi Koda, Chian-Ping Ye, Sarah C. Rogan, Andrew C. Adams, Daniel Cusher, Eleftheria Maratos–Flier, Bryan L. Roth, Bradford B. Lowell - Journal of Clinical Investigation 2011 被引用: 1,612
- Synthon-based ligand discovery in virtual libraries of over 11 billion compounds
著者: Arman A. Sadybekov, Anastasiia Sadybekov, Yongfeng Liu, Christos Iliopoulos‐Tsoutsouvas, Xi‐Ping Huang, Julie E. Pickett, Blake Houser, Nilkanth Patel, Ngan K. Tran, Fei Tong, Nikolai Zvonok, Manish K. Jain, Olena Savych, Dmytro S. Radchenko, Spyros P. Nikas, Nicos A. Petasis, Yurii S. Moroz, Bryan L. Roth, Alexandros Makriyannis, Vsevolod Katritch - Nature 2021 被引用: 433
- The Expanded Biology of Serotonin
著者: Miles Berger, J.A. Gray, Bryan L. Roth - Annual Review of Medicine 2009 被引用: 2,066
- Evolving the lock to fit the key to create a family of G protein-coupled receptors potently activated by an inert ligand
著者: Blaine N. Armbruster, Xiang Li, Mark H. Pausch, Stefan Herlitze, Bryan L. Roth - National Academy of Sciences, Proceedings of the National Academy of Sciences 2007 被引用: 2,112
- TRUPATH, an open-source biosensor platform for interrogating the GPCR transducerome
著者: Reid H. J. Olsen, Jeffrey F. DiBerto, Justin G. English, Alexis M. Glaudin, B. Krumm, Samuel T. Slocum, Tao Che, Ariana C. Gavin, John D. McCorvy, Bryan L. Roth, Ryan T. Strachan - Nature Chemical Biology 2020 被引用: 569
- PRESTO-Tango as an open-source resource for interrogation of the druggable human GPCRome
著者: Wesley K. Kroeze, Maria F. Sassano, Xi‐Ping Huang, Katherine Lansu, John D. McCorvy, Patrick M. Giguère, Noah Sciaky, Bryan L. Roth - Nature Structural & Molecular Biology 2015 被引用: 785
- Structure of a Hallucinogen-Activated Gq-Coupled 5-HT2A Serotonin Receptor
著者: Kuglae Kim, Tao Che, Ouliana Panova, Jeffrey F. DiBerto, Jiankun Lyu, B. Krumm, Daniel Wacker, Michael J. Robertson, Alpay B. Seven, David E. Nichols, Brian K. Shoichet, Georgios Skiniotis, Bryan L. Roth - Cell 2020 被引用: 501
- Bespoke library docking for 5-HT2A receptor agonists with antidepressant activity
著者: Anat Levit Kaplan, Danielle N. Confair, Kuglae Kim, Ximena Barros-Álvarez, Ramona M. Rodriguiz, Yang Ying, Oh Sang Kweon, Tao Che, John D. McCorvy, David N. Kamber, James P. Phelan, Luan Carvalho Martins, Vladimir M. Pogorelov, Jeffrey F. DiBerto, Samuel T. Slocum, Xi‐Ping Huang, Manish K. Jain, Michael J. Robertson, Ouliana Panova, Alpay B. Seven, Autumn Q. Wetsel, William C. Wetsel, John J. Irwin, Georgios Skiniotis, Brian K. Shoichet, Bryan L. Roth, Jonathan A. Ellman - Nature 2022 被引用: 252
- The neural basis of psychedelic action
著者: Alex C. Kwan, David E. Olson, Katrin H. Preller, Bryan L. Roth - Nature Neuroscience 2022 被引用: 288
- Predicting new molecular targets for known drugs
著者: Michael J. Keiser, Vincent Setola, John J. Irwin, Christian Laggner, Atheir I. Abbas, Sandra J. Hufeisen, Niels Jensen, Michael B. Kuijer, Roberto C. Matos, Thuy Tran, Ryan Whaley, Richard A. Glennon, Jérôme Hert, Kelan Thomas, Douglas D. Edwards, Brian K. Shoichet, Bryan L. Roth - Nature 2009 被引用: 1,714
- Structure-based discovery of opioid analgesics with reduced side effects
著者: Aashish Manglik, Henry Lin, Dipendra K. Aryal, John D. McCorvy, Daniela Dengler, Gregory Corder, Anat Levit, Ralf C. Kling, Viachaslau Bernat, Harald Hübner, Xi-Ping Huang, Maria F. Sassano, Patrick M. Giguère, Stefan Löber, Da Duan, Grégory Scherrer, Brian K. Kobilka, Peter Gmeiner, Bryan L. Roth, Brian K. Shoichet - Nature, Nat. 2016 被引用: 972
- Virtual discovery of melatonin receptor ligands to modulate circadian rhythms
著者: Reed M. Stein, Hye Jin Kang, John D. McCorvy, Grant C. Glatfelter, Anthony Jones, Tao Che, Samuel T. Slocum, Xi‐Ping Huang, Olena Savych, Yurii S. Moroz, Benjamin Stauch, Linda C. Johansson, Vadim Cherezov, Terry Kenakin, John J. Irwin, Brian K. Shoichet, Bryan L. Roth, Margarita L. Dubocovich - Nature 2020 被引用: 317
- Structures of the entire human opioid receptor family
著者: Yue Wang, Youwen Zhuang, Jeffrey F. DiBerto, X. Edward Zhou, Gavin P. Schmitz, Qingning Yuan, Manish K. Jain, Weiyi Liu, Karsten Melcher, Yi Jiang, Bryan L. Roth, H. Eric Xu - Cell 2023 被引用: 200
- AlphaFold2 structures guide prospective ligand discovery
著者: Jiankun Lyu, Nicholas J. Kapolka, Ryan H. Gumpper, Assaf Alon, Liang Wang, Manish K. Jain, Ximena Barros-Álvarez, Kensuke Sakamoto, Yoojoong Kim, Jeffrey F. DiBerto, Kuglae Kim, Isabella Glenn, Tia A. Tummino, Sijie Huang, John J. Irwin, Olga O. Tarkhanova, Yurii S. Moroz, Georgios Skiniotis, Andrew C. Kruse, Brian K. Shoichet, Bryan L. Roth - Science 2024 被引用: 140
- Automated design of ligands to polypharmacological profiles
著者: Jérémy Besnard, G.F. Ruda, Vincent Setola, Keren Abecassis, Ramona M. Rodriguiz, Xi‐Ping Huang, Suzanne Norval, Maria F. Sassano, Antony I. Shin, Lauren Webster, Frederick R. C. Simeons, Laste Stojanovski, Annik Prat, Nabil G. Seidah, Daniel B. Constam, G. Richard Bickerton, Kevin D. Read, William C. Wetsel, Ian H. Gilbert, Bryan L. Roth, Andrew L. Hopkins - Nature 2012 被引用: 854
- The promises and perils of psychedelic pharmacology for psychiatry
著者: Tristan McClure‐Begley, Bryan L. Roth - Nature Reviews Drug Discovery 2022 被引用: 193
- Community guidelines for GPCR ligand bias: IUPHAR review 32
著者: Peter Kolb, Terry Kenakin, S P H Alexander, Marcel Bermúdez, Laura Bohn, Christian S. Breinholt, Michel Bouvier, Stephen J. Hill, Evi Kostenis, Kirill A. Martemyanov, Rick R. Neubig, H. Ongun Onaran, Sudarshan Rajagopal, Bryan L. Roth, Jana Selent, Arun K. Shukla, M. Sommer, David E. Gloriam - British Journal of Pharmacology 2022 被引用: 222
- Crystal Structure of an LSD-Bound Human Serotonin Receptor
著者: Daniel Wacker, Sheng Wang, John D. McCorvy, Robin M. Betz, AJ Venkatakrishnan, Anat Levit, Katherine Lansu, Zachary L. Schools, Tao Che, David E. Nichols, Brian K. Shoichet, Ron O. Dror, Bryan L. Roth - Cell 2017 被引用: 472
- Structures of the σ2 receptor enable docking for bioactive ligand discovery
著者: Assaf Alon, Jiankun Lyu, João M. Bráz, Tia A. Tummino, Veronica Craik, Matthew J. O’Meara, Chase M. Webb, Dmytro S. Radchenko, Yurii S. Moroz, Xi‐Ping Huang, Yongfeng Liu, Bryan L. Roth, John J. Irwin, Allan I. Basbaum, Brian K. Shoichet, Andrew C. Kruse - Nature 2021 被引用: 194
- Remote Control of Neuronal Activity in Transgenic Mice Expressing Evolved G Protein-Coupled Receptors
著者: Georgia M. Alexander, Sarah C. Rogan, Atheir I. Abbas, Blaine N. Armbruster, Ying Pei, John Allen, Randal J. Nonneman, John F. Hartmann, Sheryl S. Moy, Miguel A. L. Nicolelis, James O McNamara, Bryan L. Roth - Neuron 2009 被引用: 1,023
- Structural insights into the human D1 and D2 dopamine receptor signaling complexes
著者: Youwen Zhuang, Peiyu Xu, Chunyou Mao, Lei Wang, B. Krumm, X. Edward Zhou, Sijie Huang, Heng Liu, Xi Cheng, Xi‐Ping Huang, Dandan Shen, Ting-Hai Xu, Yongfeng Liu, Yue Wang, Jia Guo, Yi Jiang, Hualiang Jiang, Karsten Melcher, Bryan L. Roth, Yan Zhang, Cheng Zhang, H. Eric Xu - Cell 2021 被引用: 264
- The promise and peril of chemical probes
著者: C.H. Arrowsmith, James E. Audia, Christopher P. Austin, Jonathan B. Baell, Jonathan P. Bennett, Julian Blagg, C. Bountra, Paul E. Brennan, Peter J. Brown, Mark E. Bunnage, Carolyn Buser‐Doepner, Robert M Campbell, Adrian J. Carter, Philip Cohen, Robert A. Copeland, Ben Cravatt, Jayme L. Dahlin, Dashyant Dhanak, A.M. Edwards, Mathias Frederiksen, Stephen V. Frye, Nathanael S. Gray, Charles E. Grimshaw, David Hepworth, Trevor Howe, K. Huber, Jian Jin, Stefan Knapp, Joanne Kotz, Ryan G. Kruger, Derek Lowe, Mary M. Mader, Brian D. Marsden, Anke Mueller‐Fahrnow, Susanne Müller, Rónán C. O’Hagan, John P. Overington, Dafydd R. Owen, Saul H. Rosenberg, Ruth A. Ross, Bryan L. Roth, Matthieu Schapira, Stuart L. Schreiber, Brian K. Shoichet, M. Sundström, Giulio Superti-Furga, Jack Taunton, Leticia Toledo‐Sherman, Chris Walpole, Michael A. Walters, Timothy M. Willson, Paul Workman, Robert N. Young, William J. Zuercher - Nature Chemical Biology 2015 被引用: 850
