Xi‐Ping Huang
1992–2025 年に発表
- 別表記
- Xi-Ping Huang
- 104
- 論文数
- 25,272
- 被引用数
- 72
- h 指数
- 101
- i10 指数
被引用数
引用元
国・地域
機関
分野
- Biochemistry, Genetics and Molecular Biology33.3%
- Medicine31.1%
- Neuroscience13.6%
- Computer Science10%
- Immunology and Microbiology3.3%
- Psychology2.2%
- その他6.5%
トピック
- Receptor Mechanisms and Signaling6.6%
- Computational Drug Discovery Methods5.6%
- SARS-CoV-2 and COVID-19 Research4.9%
- Neuropeptides and Animal Physiology3.6%
- COVID-19 Clinical Research Studies3.1%
- Neuroscience and Neuropharmacology Research3%
- その他73.2%
共著者
- Bryan L. Roth74
- Brian K. Shoichet16
- Jian Jin16
- John D. McCorvy16
- Vsevolod Katritch15
- Yongfeng Liu15
- B. Krumm12
- Samuel T. Slocum11
- Vadim Cherezov11
- Jeffrey F. DiBerto10
- Raymond C. Stevens10
- Tao Che9
- Gye Won Han8
- Jonathan F. Fay8
- Vincent Setola8
- Jing Liu7
- John J. Irwin7
- Reid H. J. Olsen7
- Daniel Wacker6
- Eyal Vardy6
- Hye Jin Kang6
- Marc G. Caron6
- Peter J. Brown6
- Stephen V. Frye6
全論文
- A SARS-CoV-2 protein interaction map reveals targets for drug repurposing
著者: David E. Gordon, Gwendolyn Μ. Jang, Mehdi Bouhaddou, Jiewei Xu, Kirsten Obernier, Kris M. White, Matthew J. O’Meara, Veronica V. Rezelj, Jeffrey Guo, Danielle L. Swaney, Tia A. Tummino, Ruth Hüttenhain, Robyn M. Kaake, Alicia Richards, Beril Tutuncuoglu, Helene Foussard, Jyoti Batra, Kelsey M. Haas, Maya Modak, Minkyu Kim, Paige Haas, Benjamin J. Polacco, Hannes Braberg, Jacqueline M. Fabius, Manon Eckhardt, Margaret Soucheray, Melanie J. Bennett, Merve Çakır, Michael McGregor, Qiongyu Li, Bjoern Meyer, Ferdinand Roesch, Thomas Vallet, Alice Mac Kain, Lisa Miorin, Elena Moreno, Zun Zar Chi Naing, Yuan Zhou, Shiming Peng, Ying Shi, Ziyang Zhang, Wenqi Shen, Ilsa T. Kirby, James E. Melnyk, John S. Chorba, Kevin Lou, Shizhong Dai, Inigo Barrio‐Hernandez, Danish Memon, Claudia Hernández-Armenta, Jiankun Lyu, Christopher J.P. Mathy, Tina Perica, Kala Bharath Pilla, Sai J. Ganesan, Daniel J. Saltzberg, Ramachandran Rakesh, Liu Xi, Sara B. Rosenthal, Lorenzo Calviello, Srivats Venkataramanan, José Liboy-Lugo, Yizhu Lin, Xi‐Ping Huang, Yongfeng Liu, Stephanie A. Wankowicz, Markus‐Frederik Bohn, Maliheh Safari, Fatima S. Ugur, Cassandra Koh, Nastaran Sadat Savar, Quang Tran, Djoshkun Shengjuler, Sabrina Johanna Fletcher, Michael C. O’Neal, Yiming Cai, Jason C. Chang, David Broadhurst, Saker Klippsten, Phillip P. Sharp, Nicole A. Wenzell, Duygu Kuzuoğlu‐Öztürk, Hao‐Yuan Wang, Raphael Trenker, Janet M. Young, Devin A. Cavero, Joseph Hiatt, Theodore L. Roth, Ujjwal Rathore, Advait Subramanian, Julia Noack, Mathieu Hubert, Robert M. Stroud, Alan D. Frankel, Oren S. Rosenberg, Kliment A. Verba, David A. Agard, Mélanie Ott, Michael Emerman, Natalia Jura ほか 25 名 - Nature 2020 被引用: 4,888
- Synthon-based ligand discovery in virtual libraries of over 11 billion compounds
著者: Arman A. Sadybekov, Anastasiia Sadybekov, Yongfeng Liu, Christos Iliopoulos‐Tsoutsouvas, Xi‐Ping Huang, Julie E. Pickett, Blake Houser, Nilkanth Patel, Ngan K. Tran, Fei Tong, Nikolai Zvonok, Manish K. Jain, Olena Savych, Dmytro S. Radchenko, Spyros P. Nikas, Nicos A. Petasis, Yurii S. Moroz, Bryan L. Roth, Alexandros Makriyannis, Vsevolod Katritch - Nature 2021 被引用: 433
- NMDAR inhibition-independent antidepressant actions of ketamine metabolites
著者: Panos Zanos, Ruin Moaddel, Patrick J. Morris, Polymnia Georgiou, Jonathan Fischell, Gregory I. Elmer, Manickavasagom Alkondon, Peixiong Yuan, Heather J. Pribut, N. Singh, Katina S. S. Dossou, Yuhong Fang, Xi‐Ping Huang, Cheryl L. Mayo, Irving W. Wainer, Edson X. Albuquerque, Scott M. Thompson, Craig J. Thomas, Carlos A. Zarate, Todd D. Gould - Nature 2016 被引用: 1,619
- PRESTO-Tango as an open-source resource for interrogation of the druggable human GPCRome
著者: Wesley K. Kroeze, Maria F. Sassano, Xi‐Ping Huang, Katherine Lansu, John D. McCorvy, Patrick M. Giguère, Noah Sciaky, Bryan L. Roth - Nature Structural & Molecular Biology 2015 被引用: 785
- Bespoke library docking for 5-HT2A receptor agonists with antidepressant activity
著者: Anat Levit Kaplan, Danielle N. Confair, Kuglae Kim, Ximena Barros-Álvarez, Ramona M. Rodriguiz, Yang Ying, Oh Sang Kweon, Tao Che, John D. McCorvy, David N. Kamber, James P. Phelan, Luan Carvalho Martins, Vladimir M. Pogorelov, Jeffrey F. DiBerto, Samuel T. Slocum, Xi‐Ping Huang, Manish K. Jain, Michael J. Robertson, Ouliana Panova, Alpay B. Seven, Autumn Q. Wetsel, William C. Wetsel, John J. Irwin, Georgios Skiniotis, Brian K. Shoichet, Bryan L. Roth, Jonathan A. Ellman - Nature 2022 被引用: 252
- Structure-based discovery of opioid analgesics with reduced side effects
著者: Aashish Manglik, Henry Lin, Dipendra K. Aryal, John D. McCorvy, Daniela Dengler, Gregory Corder, Anat Levit, Ralf C. Kling, Viachaslau Bernat, Harald Hübner, Xi-Ping Huang, Maria F. Sassano, Patrick M. Giguère, Stefan Löber, Da Duan, Grégory Scherrer, Brian K. Kobilka, Peter Gmeiner, Bryan L. Roth, Brian K. Shoichet - Nature, Nat. 2016 被引用: 972
- Virtual discovery of melatonin receptor ligands to modulate circadian rhythms
著者: Reed M. Stein, Hye Jin Kang, John D. McCorvy, Grant C. Glatfelter, Anthony Jones, Tao Che, Samuel T. Slocum, Xi‐Ping Huang, Olena Savych, Yurii S. Moroz, Benjamin Stauch, Linda C. Johansson, Vadim Cherezov, Terry Kenakin, John J. Irwin, Brian K. Shoichet, Bryan L. Roth, Margarita L. Dubocovich - Nature 2020 被引用: 317
- Automated design of ligands to polypharmacological profiles
著者: Jérémy Besnard, G.F. Ruda, Vincent Setola, Keren Abecassis, Ramona M. Rodriguiz, Xi‐Ping Huang, Suzanne Norval, Maria F. Sassano, Antony I. Shin, Lauren Webster, Frederick R. C. Simeons, Laste Stojanovski, Annik Prat, Nabil G. Seidah, Daniel B. Constam, G. Richard Bickerton, Kevin D. Read, William C. Wetsel, Ian H. Gilbert, Bryan L. Roth, Andrew L. Hopkins - Nature 2012 被引用: 854
- Structures of the σ2 receptor enable docking for bioactive ligand discovery
著者: Assaf Alon, Jiankun Lyu, João M. Bráz, Tia A. Tummino, Veronica Craik, Matthew J. O’Meara, Chase M. Webb, Dmytro S. Radchenko, Yurii S. Moroz, Xi‐Ping Huang, Yongfeng Liu, Bryan L. Roth, John J. Irwin, Allan I. Basbaum, Brian K. Shoichet, Andrew C. Kruse - Nature 2021 被引用: 194
- Structural insights into the human D1 and D2 dopamine receptor signaling complexes
著者: Youwen Zhuang, Peiyu Xu, Chunyou Mao, Lei Wang, B. Krumm, X. Edward Zhou, Sijie Huang, Heng Liu, Xi Cheng, Xi‐Ping Huang, Dandan Shen, Ting-Hai Xu, Yongfeng Liu, Yue Wang, Jia Guo, Yi Jiang, Hualiang Jiang, Karsten Melcher, Bryan L. Roth, Yan Zhang, Cheng Zhang, H. Eric Xu - Cell 2021 被引用: 264
- Structure, function and pharmacology of human itch GPCRs
著者: Can Cao, Hye Jin Kang, Isha Singh, He Chen, Chengwei Zhang, Wenlei Ye, Byron W. Hayes, Jing Liu, Ryan H. Gumpper, Brian J. Bender, Samuel T. Slocum, B. Krumm, Katherine Lansu, John D. McCorvy, Wesley K. Kroeze, Justin G. English, Jeffrey F. DiBerto, Reid H. J. Olsen, Xi‐Ping Huang, Shicheng Zhang, Yongfeng Liu, Kuglae Kim, Joel Karpiak, Lily Yeh Jan, Soman N. Abraham, Jian Jin, Brian K. Shoichet, Jonathan F. Fay, Bryan L. Roth - Nature 2021 被引用: 224
- Structure-based discovery of nonopioid analgesics acting through the α 2A -adrenergic receptor
著者: Elissa A. Fink, Jun Xu, Harald Hübner, João M. Bráz, Philipp Seemann, Charlotte Avet, Veronica Craik, Dorothée Weikert, Maximilian F. Schmidt, Chase M. Webb, Nataliya A. Tolmachova, Yurii S. Moroz, Xi‐Ping Huang, Chakrapani Kalyanaraman, Stefan Gahbauer, Geng Chen, Zheng Liu, Matthew P. Jacobson, John J. Irwin, Michel Bouvier, Yang Du, Brian K. Shoichet, Allan I. Basbaum, Peter Gmeiner - Science 2022 被引用: 152
- Discovery of Human Signaling Systems: Pairing Peptides to G Protein-Coupled Receptors
著者: Simon R. Foster, Alexander S. Hauser, Line Vedel, Ryan T. Strachan, Xi‐Ping Huang, Ariana C. Gavin, Sushrut D. Shah, Ajay P. Nayak, Linda M. Haugaard‐Kedström, Raymond B. Penn, Bryan L. Roth, Hans Bräuner‐Osborne, David E. Gloriam - Cell 2019 被引用: 267
- Structure-based discovery of conformationally selective inhibitors of the serotonin transporter
著者: Isha Singh, Anubha Seth, Christian B. Billesbølle, João M. Bráz, Ramona M. Rodriguiz, Kasturi Roy, Bethlehem Bekele, Veronica Craik, Xi‐Ping Huang, Danila Boytsov, Vladimir M. Pogorelov, Parnian Lak, Henry O’Donnell, Walter Sandtner, John J. Irwin, Bryan L. Roth, Allan I. Basbaum, William C. Wetsel, Aashish Manglik, Brian K. Shoichet, Gary Rudnick - Cell 2023 被引用: 99
- Allosteric ligands for the pharmacologically dark receptors GPR68 and GPR65
著者: Xi-Ping Huang, Joel Karpiak, Wesley K. Kroeze, Hu Zhu, Xin Chen, Sheryl S. Moy, Kara A. Saddoris, Viktoriya D. Nikolova, Martilias S. Farrell, Sheng Wang, Thomas J. Mangano, Deepak A. Deshpande, Alice Jiang, Raymond B. Penn, Jian Jin, Beverly H. Koller, Terry Kenakin, Brian K. Shoichet, Bryan L. Roth - Nature, Nat. 2015 被引用: 287
- Structure of the human κ-opioid receptor in complex with JDTic
著者: Huixian Wu, Daniel Wacker, Mauro Mileni, Vsevolod Katritch, Gye Won Han, Eyal Vardy, Wei Liu, Aaron A. Thompson, Xi‐Ping Huang, F. Ivy Carroll, S. Wayne Mascarella, Richard B. Westkaemper, Philip D. Mosier, Bryan L. Roth, Vadim Cherezov, Raymond C. Stevens - Nature 2012 被引用: 878
- A chemical probe selectively inhibits G9a and GLP methyltransferase activity in cells
著者: Masoud Vedadi, Dalia Baršytė-Lovejoy, Feng Liu, Sylvie Rival‐Gervier, Abdellah Allali‐Hassani, Viviane Labrie, Tim J. Wigle, Peter A. DiMaggio, Gregory A. Wasney, Alena Siarheyeva, Aiping Dong, W. Tempel, Sun-Chong Wang, Xin Chen, Irene Chau, Thomas J Mangano, Xi‐Ping Huang, Catherine Simpson, Samantha G Pattenden, Jacqueline L Norris, Dmitri Kireev, Ashutosh Tripathy, A.M. Edwards, Bryan L. Roth, William P Janzen, Benjamin A. García, Artūras Petronis, James Ellis, Peter J. Brown, Stephen V. Frye, C.H. Arrowsmith, Jian Jin - Nature Chemical Biology 2011 被引用: 531
- Structure of the Nanobody-Stabilized Active State of the Kappa Opioid Receptor
著者: Tao Che, Susruta Majumdar, Saheem A. Zaidi, Pauline W. Ondachi, John D. McCorvy, Sheng Wang, Philip D. Mosier, Rajendra Uprety, Eyal Vardy, B. Krumm, Gye Won Han, Ming-Yue Lee, Els Pardon, Jan Steyaert, Xi‐Ping Huang, Ryan T. Strachan, Alexandra R. Tribo, Gavril W. Pasternak, F. Ivy Carroll, Raymond C. Stevens, Vadim Cherezov, Vsevolod Katritch, Daniel Wacker, Bryan L. Roth - Cell 2018 被引用: 377
- Molecular control of δ-opioid receptor signalling
著者: Gustavo Fenalti, Patrick M. Giguère, Vsevolod Katritch, Xi‐Ping Huang, Aaron A. Thompson, Vadim Cherezov, Bryan L. Roth, Raymond C. Stevens - Nature 2014 被引用: 503
- An Orally Bioavailable Chemical Probe of the Lysine Methyltransferases EZH2 and EZH1
著者: Kyle D. Konze, Anqi Ma, Fengling Li, Dalia Baršytė-Lovejoy, Trevor Parton, Christopher J. MacNevin, Feng Liu, Cen Gao, Xi‐Ping Huang, Ekaterina Kuznetsova, Marie Rougié, Alice Jiang, Samantha G. Pattenden, Jacqueline L. Norris, Lindsey I. James, Bryan L. Roth, Peter J. Brown, Stephen V. Frye, C.H. Arrowsmith, Klaus M. Hahn, Gang Greg Wang, Masoud Vedadi, Jian Jin - ACS Chemical Biology 2013 被引用: 466
- A New DREADD Facilitates the Multiplexed Chemogenetic Interrogation of Behavior
著者: Eyal Vardy, J. Elliott Robinson, Chia Li, Reid H. J. Olsen, Jeffrey F. DiBerto, Patrick M. Giguère, Flori M. Sassano, Xi‐Ping Huang, Hu Zhu, Daniel J. Urban, Kate White, Joseph E. Rittiner, Nicole A. Crowley, Kristen E. Pleil, Christopher M. Mazzone, Philip D. Mosier, Juan Song, Thomas L. Kash, C. J. Malanga, Michael J. Krashes, Bryan L. Roth - Neuron 2015 被引用: 398
- Mechanism of dopamine binding and allosteric modulation of the human D1 dopamine receptor
著者: Youwen Zhuang, B. Krumm, Huibing Zhang, X. Edward Zhou, Yue Wang, Xi‐Ping Huang, Yongfeng Liu, Xi Cheng, Yi Jiang, Hualiang Jiang, Cheng Zhang, Wei Yi, Bryan L. Roth, Yan Zhang, H. Eric Xu - Cell Research 2021 被引用: 99
- Neurotensin Receptor Allosterism Revealed in Complex with a Biased Allosteric Modulator
著者: B. Krumm, Jeffrey F. DiBerto, Reid H. J. Olsen, Hye Jin Kang, Samuel T. Slocum, Shicheng Zhang, Ryan T. Strachan, Xi‐Ping Huang, Lauren M. Slosky, Anthony B. Pinkerton, Lawrence S Barak, Marc G. Caron, Terry Kenakin, Jonathan F. Fay, Bryan L. Roth - Biochemistry 2023 被引用: 71
- A Simple Representation of Three-Dimensional Molecular Structure
著者: Seth D. Axen, Xi‐Ping Huang, Elena L. Cáceres, Leo Gendelev, Bryan L. Roth, Michael J. Keiser - Journal of Medicinal Chemistry 2017 被引用: 146
